SCHEMBL6141563

SCHEMBL6141563

O=C(O)C(Cc1ccc2nc(-c3c(F)cccc3Cl)ccc2c1)[AsH]C(=O)C1(c2ccc(Cl)cc2)CCCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 3/20 0.46
ITGAV P06756 1/20 0.46
ABL1 P00519 1/20 0.34
TRPA1 O75762 4/20 0.33
HDAC4 P56524 2/20 0.33
ITGA4 P13612 2/20 0.33
CYP3A4 P08684 1/20 0.32
CYP2C8 P10632 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KCNH2 Q12809 1/20 0.32
PTPN2 P17706 2/20 0.32
PTPN1 P18031 2/20 0.32
CDC25B P30305 2/20 0.32
PTPN6 P29350 1/20 0.32
FFAR2 O15552 3/20 0.31
ITGB7 P26010 1/20 0.31
ALDH1A1 P00352 1/20 0.30
AVPR1A P37288 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6142036 0.89 ITGB1 (0.37) ITGB1ITGAVTRPA1HDAC4ITGA4
SCHEMBL3313410 0.85 ITGB1 (0.59) ITGB1ITGAVITGA4PTPN2PTPN1
SCHEMBL4624848 0.81 ITGB1 (0.54) ITGB1ITGAVITGA4PTPN2PTPN1
SCHEMBL4625262 0.79 ITGB1 (0.66) ITGB1ITGAVITGA4PTPN1ITGB7
SCHEMBL3313181 0.79 ITGB1 (0.66) ITGB1ITGAVITGA4PTPN1ITGB7
SCHEMBL6141406 0.76 ITGB1 (0.50) ITGB1ITGAVABL1ITGA4KCNH2
SCHEMBL6141402 0.76 ITGB1 (0.50) ITGB1ITGAVABL1ITGA4KCNH2
SCHEMBL6141473 0.75 ITGB1 (0.55) ITGB1ITGAVABL1ITGA4KCNH2
SCHEMBL4624559 0.74 ITGB1 (0.54) ITGB1ITGAVABL1HDAC4ITGA4
SCHEMBL3316847 0.74 ITGB1 (0.48) ITGB1ITGAVITGA4PTPN2PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2005-02-02 EP claimed
WO-2003093237-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2003-11-13 WO claimed