SCHEMBL6142122

SCHEMBL6142122

COc1ccc2c(C(=O)c3ccc(OCCN4CCCCC4)cc3)c(-c3ccccc3OC)sc2c1

nearest known ligand 0.76

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 19/20 0.76
ESR2 Q92731 19/20 0.76
ENPP3 O14638 1/20 0.64
ENPP1 P22413 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6141708 0.93 ESR1 (0.84) ESR1ESR2ENPP3ENPP1
SCHEMBL6141716 0.91 ESR1 (0.84) ESR1ESR2ENPP3ENPP1
SCHEMBL8674595 0.90 ESR1 (0.83) ESR1ESR2ENPP3ENPP1
SCHEMBL5419626 0.89 ESR1 (0.72) ESR1ESR2ENPP3ENPP1
SCHEMBL8598353 0.88 ESR1 (0.89) ESR1ESR2ENPP3ENPP1
SCHEMBL8598366 0.88 ESR1 (0.89) ESR1ESR2ENPP3ENPP1
SCHEMBL6141703 0.88 ESR1 (0.80) ESR1ESR2ENPP3ENPP1
SCHEMBL8600306 0.87 ESR1 (0.88) ESR1ESR2ENPP3ENPP1
SCHEMBL6142024 0.87 ESR1 (0.77) ESR1ESR2ENPP3ENPP1
SCHEMBL6141664 0.87 ESR1 (0.86) ESR1ESR2ENPP3ENPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1493741-A2 Benzo[b]thiophene compounds, intermediates, processes, compositions and methods Eli Lilly & Company (US) 2005-01-05 EP disclosed
EP-0826683-B1 Benzo[B]thiophene compounds, intermediates, processes, compositions, and methods LILLY CO ELI (US) 2004-10-06 EP disclosed
US-5998442-A ANTICHOLESTEROL AGENTS ELI LILLY AND COMPANY (US) 1999-12-07 US disclosed
EP-0826683-A1 Benzo[B]thiophene compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 1998-03-04 EP disclosed