SCHEMBL6142673

SCHEMBL6142673

COC(=O)C(Cc1ccc2nc(-c3c(Cl)cccc3Cl)ccc2c1)[AsH]C(=O)OC(C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 5/20 0.52
ITGAV P06756 1/20 0.52
ABL1 P00519 1/20 0.37
ITGA4 P13612 4/20 0.33
ITGB7 P26010 3/20 0.33
DGAT1 O75907 1/20 0.33
CTSB P07858 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
CTSL P07711 1/20 0.31
CDK2 P24941 1/20 0.31
TACR3 P29371 1/20 0.30
HRH3 Q9Y5N1 3/20 0.30
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30
MAPT P10636 1/20 0.30
KCNH2 Q12809 2/20 0.30
THRB P10828 1/20 0.30
LCK P06239 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6141061 0.91 ITGB1 (0.55) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL6141998 0.89 ITGB1 (0.39) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL3320795 0.83 ITGB1 (0.59) ITGB1ITGAVITGA4ITGB7CTSB
SCHEMBL4627521 0.83 ITGB1 (0.59) ITGB1ITGAVITGA4ITGB7CTSB
SCHEMBL1030225 0.83 ITGB1 (0.59) ITGB1ITGAVITGA4ITGB7CTSB
SCHEMBL6141873 0.81 ITGB1 (0.53) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL3321001 0.80 ITGB1 (0.60) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL3313415 0.80 ITGB1 (0.59) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL4750010 0.80 ITGB1 (0.59) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL6141516 0.79 ITGB1 (0.51) ITGB1ITGAVITGA4ITGB7MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2005-02-02 EP claimed
WO-2003093237-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2003-11-13 WO claimed