SCHEMBL6141516

SCHEMBL6141516

COC(=O)C(Cc1ccc2nc(-c3c(OC)cccc3OC)ccc2c1)[AsH]C(=O)c1c(Cl)cccc1Cl

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 14/20 0.51
ITGAV P06756 1/20 0.51
ITGA4 P13612 16/20 0.39
ITGB7 P26010 12/20 0.35
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6140931 0.92 ITGB1 (0.54) ITGB1ITGAVITGA4ITGB7
SCHEMBL6141873 0.89 ITGB1 (0.53) ITGB1ITGAVITGA4ITGB7
SCHEMBL6140590 0.85 ITGB1 (0.56) ITGB1ITGAVITGA4ITGB7
SCHEMBL6141998 0.83 ITGB1 (0.39) ITGB1ITGAVITGA4ITGB7
SCHEMBL3313321 0.83 ITGB1 (0.69) ITGB1ITGAVITGA4ITGB7
SCHEMBL4627302 0.83 ITGB1 (0.69) ITGB1ITGAVITGA4ITGB7
SCHEMBL6142370 0.81 ITGB1 (0.66) ITGB1ITGAVITGA4ITGB7
SCHEMBL3318793 0.79 ITGB1 (0.81) ITGB1ITGAVITGA4ITGB7
SCHEMBL6142673 0.79 ITGB1 (0.52) ITGB1ITGAVITGA4ITGB7MAPT
SCHEMBL3314866 0.79 ITGB1 (0.81) ITGB1ITGAVITGA4ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2005-02-02 EP disclosed
WO-2003093237-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2003-11-13 WO disclosed