SCHEMBL6142909

SCHEMBL6142909

O[C@@H]1CN[C@H](c2ccccc2)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.46
PRCP P42785 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
PARP3 Q9Y6F1 1/20 0.37
SCN10A Q9Y5Y9 1/20 0.36
MAOA P21397 5/20 0.35
MAOB P27338 5/20 0.35
KDM1A O60341 4/20 0.35
CYP2C19 P33261 4/20 0.35
CYP2B6 P20813 3/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C9 P11712 2/20 0.35
LMNA P02545 1/20 0.35
CYP3A4 P08684 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA2A P08913 1/20 0.35
CYP2A6 P11509 1/20 0.35
SLC6A2 P23975 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5739415 1.00 GBA1 (0.46) GBA1PRCPMEN1KMT2APARP3
SCHEMBL24365777 0.82 GBA1 (0.44) GBA1PRCPMEN1KMT2APARP3
SCHEMBL29081640 0.82 GBA1 (0.44) GBA1PRCPMEN1KMT2APARP3
SCHEMBL24367023 0.82 GBA1 (0.44) GBA1PRCPMEN1KMT2APARP3
SCHEMBL8565971 0.80 SCN10A (0.38) PRCPSCN10ACYP2C19CYP1A2HSD17B10
SCHEMBL4685465 0.80 CDC7 (0.40) SCN10AMAOBKDM1ACYP2C19CYP2D6
SCHEMBL27603362 0.80 SCN10A (0.35) MEN1KMT2ASCN10ACYP3A4HSD17B10
SCHEMBL4195137 0.80 SLC18A3 (0.39) GBA1PRCPMEN1KMT2ACYP2C19
SCHEMBL24365527 0.80 SLC18A3 (0.39) GBA1PRCPMEN1KMT2ACYP2C19
SCHEMBL9158920 0.80 SLC18A3 (0.39) GBA1PRCPMEN1KMT2ACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1515949-B1 MITOTIC KINESIN INHIBITORS MERCK & CO INC (US) 2007-03-14 EP disclosed
EP-1515949-A4 MITOTIC KINESIN INHIBITORS MERCK & CO INC (US) 2005-11-09 EP disclosed
EP-1515724-A4 MITOTIC KINESIN INHIBITORS MERCK & CO INC (US) 2005-08-17 EP disclosed
EP-1515724-A1 MITOTIC KINESIN INHIBITORS Merck & Co., Inc. (US) 2005-03-23 EP disclosed
EP-1515949-A1 MITOTIC KINESIN INHIBITORS Merck & Co., Inc. (US) 2005-03-23 EP disclosed
WO-2004087050-A2 MITOTIC KINESIN INHIBITORS MERCK & CO., INC. (US) 2004-10-14 WO disclosed
WO-2003106417-A1 MITOTIC KINESIN INHIBITORS MERCK & CO., INC. (US) 2003-12-24 WO disclosed
WO-2003105855-A1 MITOTIC KINESIN INHIBITORS MERCK & CO., INC. (US) 2003-12-24 WO disclosed