SCHEMBL6146451

SCHEMBL6146451

CCCCCC(C=Cc1ccc(C(=O)O)cc1)c1ccc2c(c1)C(C)(C)CCO2

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RARA P10276 9/20 0.54
RARB P10826 9/20 0.54
RARG P13631 9/20 0.54
RXRA P19793 5/20 0.44
HNF4A P41235 2/20 0.44
SSTR5 P35346 2/20 0.41
CYP26A1 O43174 1/20 0.40
CYP26B1 Q9NR63 1/20 0.40
RXRB P28702 1/20 0.39
STAT3 P40763 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6147473 1.00 RARA (0.54) RARARARBRARGRXRAHNF4A
SCHEMBL6147479 1.00 RARA (0.54) RARARARBRARGRXRAHNF4A
SCHEMBL6146448 1.00 RARA (0.54) RARARARBRARGRXRAHNF4A
SCHEMBL4850319 0.93 RARB (0.50) RARARARBRARGRXRAHNF4A
SCHEMBL4850323 0.93 RARB (0.50) RARARARBRARGRXRAHNF4A
SCHEMBL4850328 0.93 RARB (0.50) RARARARBRARGRXRAHNF4A
SCHEMBL6146781 0.90 RARB (0.47) RARARARBRARGRXRAHNF4A
SCHEMBL6146777 0.90 RARB (0.47) RARARARBRARGRXRAHNF4A
SCHEMBL6146779 0.90 RARB (0.47) RARARARBRARGRXRAHNF4A
SCHEMBL6146774 0.90 RARB (0.47) RARARARBRARGRXRAHNF4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020026060-A1 RAR selective retinoid agonists F.HOFFMANN-LA ROCHE AG (CH) 2002-02-28 US claimed
EP-1280757-B1 NEW GAMMA SELECTIVE RETINOIDS HOFFMANN LA ROCHE (CH) 2005-08-17 EP disclosed
US-6603012-B2 RAR selective retinoid agonists HOFFMANN-LA ROCHE INC. 2003-08-05 US disclosed
EP-1280757-A2 NEW GAMMA SELECTIVE RETINOIDS F. HOFFMANN-LA ROCHE AG (CH) 2003-02-05 EP disclosed
US-20020026060-A1 RAR selective retinoid agonists F.HOFFMANN-LA ROCHE AG (CH) 2002-02-28 US disclosed
WO-2001083438-A2 NEW GAMMA SELECTIVE RETINOIDS F. HOFFMANN-LA ROCHE AG (CH) 2001-11-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020026060-A1 RAR selective retinoid agonists RARA, RARG, RARB RARA 1/4885RARB 3/4885RARG 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.