SCHEMBL6150477

SCHEMBL6150477

COC(=O)[C@H](CCC(=O)N1CCC(Cn2cccc2)CC1)NC(=O)[C@@H]1CCCN1S(=O)(=O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 19/20 0.47
ITGA4 P13612 19/20 0.47
ITGB7 P26010 2/20 0.45
HCRTR1 O43613 1/20 0.42
HCRTR2 O43614 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6150480 1.00 ITGB1 (0.47) ITGB1ITGA4ITGB7HCRTR1HCRTR2
SCHEMBL6403268 0.91 ITGB1 (0.51) ITGB1ITGA4ITGB7
SCHEMBL6403264 0.91 ITGB1 (0.51) ITGB1ITGA4ITGB7
SCHEMBL6156385 0.86 ITGB1 (0.45) ITGB1ITGA4ITGB7HCRTR1HCRTR2
SCHEMBL6156389 0.86 ITGB1 (0.45) ITGB1ITGA4ITGB7HCRTR1HCRTR2
SCHEMBL6158937 0.84 ITGB1 (0.46) ITGB1ITGA4ITGB7HCRTR1HCRTR2
SCHEMBL6151159 0.84 ITGB1 (0.46) ITGB1ITGA4ITGB7HCRTR1HCRTR2
SCHEMBL6158932 0.84 ITGB1 (0.46) ITGB1ITGA4ITGB7HCRTR1HCRTR2
SCHEMBL6151156 0.84 ITGB1 (0.46) ITGB1ITGA4ITGB7HCRTR1HCRTR2
SCHEMBL6157260 0.83 ITGB1 (0.45) ITGB1ITGA4ITGB7HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1495044-A1 HETEROCYCLIC AMIDES WITH ALPHA-4 INTEGRIN ANTAGONIST ACTIVITY J. Uriach y Compania S.A. (ES) 2005-01-12 EP claimed
WO-2003084984-A1 HETEROCYCLIC AMIDES WITH ALPHA-4 INTEGRIN ANTAGONIST ACTIVITY J. URIACH Y COMPANIA S.A. (ES) 2003-10-16 WO claimed