SCHEMBL6152815

SCHEMBL6152815

CCC(CC)(C(=O)O)C(=O)N1CCC(CCN2[C@@H]3CC[C@H]2CC(n2c(C)nc4ccccc42)C3)(c2cccc(F)c2)CC1

nearest known ligand 0.86

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 10/20 0.86
CCR5 P51681 12/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3526061 0.94 KCNH2 (0.85) KCNH2CCR5
SCHEMBL3530722 0.93 KCNH2 (1.00) KCNH2CCR5
SCHEMBL13543882 0.93 KCNH2 (1.00) KCNH2CCR5
SCHEMBL13543112 0.93 CCR5 (0.86) KCNH2CCR5
SCHEMBL13543829 0.92 KCNH2 (0.83) KCNH2CCR5
SCHEMBL3529449 0.92 KCNH2 (0.83) KCNH2CCR5
SCHEMBL13544261 0.92 KCNH2 (1.00) KCNH2CCR5
SCHEMBL3526647 0.92 KCNH2 (1.00) KCNH2CCR5
SCHEMBL3526001 0.91 KCNH2 (0.84) KCNH2CCR5
SCHEMBL3526013 0.90 KCNH2 (0.89) KCNH2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569646-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2005-09-07 EP disclosed
WO-2004054974-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2004-07-01 WO disclosed