SCHEMBL6153030

SCHEMBL6153030

O=C(O)C(CCC(=O)N1CCC(CCOC(=O)N2CCN(c3ccccc3)CC2)CC1)NC(=O)[C@@H]1CCCN1S(=O)(=O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 11/20 0.47
ITGB1 P05556 11/20 0.47
ITGB7 P26010 2/20 0.47
CHRM4 P08173 4/20 0.42
ITGA2 P17301 1/20 0.41
P2RY12 Q9H244 2/20 0.41
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
ITGA5 P08648 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6402915 1.00 ITGA4 (0.47) ITGA4ITGB1ITGB7CHRM4ITGA2
SCHEMBL6402913 1.00 ITGA4 (0.47) ITGA4ITGB1ITGB7CHRM4ITGA2
SCHEMBL6159009 0.92 ITGB1 (0.49) ITGA4ITGB1ITGB7
SCHEMBL6147636 0.92 ITGB1 (0.49) ITGA4ITGB1ITGB7
SCHEMBL6150353 0.92 ITGB1 (0.49) ITGA4ITGB1ITGB7
SCHEMBL6401978 0.90 ITGB1 (0.48) ITGA4ITGB1ITGB7ITGA2
SCHEMBL6149415 0.90 ITGB1 (0.48) ITGA4ITGB1ITGB7ITGA2
SCHEMBL6401982 0.90 ITGB1 (0.48) ITGA4ITGB1ITGB7ITGA2
SCHEMBL6149727 0.83 ITGA4 (0.44) ITGA4ITGB1ITGB7ITGA2ITGB3
SCHEMBL6402116 0.83 ITGA4 (0.44) ITGA4ITGB1ITGB7ITGA2ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1495044-A1 HETEROCYCLIC AMIDES WITH ALPHA-4 INTEGRIN ANTAGONIST ACTIVITY J. Uriach y Compania S.A. (ES) 2005-01-12 EP disclosed
WO-2003084984-A1 HETEROCYCLIC AMIDES WITH ALPHA-4 INTEGRIN ANTAGONIST ACTIVITY J. URIACH Y COMPANIA S.A. (ES) 2003-10-16 WO disclosed