SCHEMBL6153228

SCHEMBL6153228

Cc1nc2ccccc2n1C1C[C@H]2CC[C@@H](C1)N2CCC1(c2ccccc2)CCN(C(=O)c2cccc(C(=N)NO)c2)CC1

nearest known ligand 0.86

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 10/20 0.86
CCR5 P51681 11/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3528707 0.91 KCNH2 (1.00) KCNH2CCR5
SCHEMBL3527806 0.91 KCNH2 (1.00) KCNH2CCR5
SCHEMBL13543129 0.91 KCNH2 (1.00) KCNH2CCR5
SCHEMBL13543130 0.90 KCNH2 (1.00) KCNH2CCR5
SCHEMBL3524678 0.90 KCNH2 (1.00) KCNH2CCR5
SCHEMBL13544043 0.90 CCR5 (1.00) KCNH2CCR5
SCHEMBL13543123 0.90 CCR5 (1.00) KCNH2CCR5
SCHEMBL3523862 0.90 CCR5 (1.00) KCNH2CCR5
SCHEMBL13543577 0.90 CCR5 (1.00) KCNH2CCR5
SCHEMBL13543411 0.89 CCR5 (1.00) KCNH2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569646-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2005-09-07 EP disclosed
WO-2004054974-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2004-07-01 WO disclosed