SCHEMBL6153901

SCHEMBL6153901

O=C(O)N1C2CCC1CC(Nc1ccccc1)C2

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 8/20 0.49
OPRM1 P35372 1/20 0.48
OPRD1 P41143 1/20 0.48
OPRK1 P41145 1/20 0.48
KCNH2 Q12809 1/20 0.48
ALDH1A1 P00352 1/20 0.48
MEN1 O00255 1/20 0.43
MAPK1 P28482 1/20 0.43
KMT2A Q03164 1/20 0.43
HTT P42858 1/20 0.42
GAA P10253 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
LMNA P02545 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CHRM1 P11229 2/20 0.40
CHRM4 P08173 1/20 0.40
CHRM5 P08912 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7460238 0.81 KMT2A (0.54) OPRM1OPRD1OPRK1KCNH2MAPK1
SCHEMBL7226906 0.80 GAA (0.50) LTA4HOPRM1OPRD1OPRK1KCNH2
SCHEMBL7237208 0.80 GAA (0.50) LTA4HOPRM1OPRD1OPRK1KCNH2
SCHEMBL4396685 0.80 GAA (0.50) LTA4HOPRM1OPRD1OPRK1KCNH2
SCHEMBL3524222 0.80 CHRM1 (0.55) LTA4HALDH1A1MAPK1KMT2AHTT
SCHEMBL7464902 0.77 CHRM4 (0.54) OPRM1OPRD1OPRK1KCNH2MEN1
SCHEMBL1574043 0.76 MEN1 (0.55) MEN1MAPK1KMT2AGAACHRM1
SCHEMBL21773167 0.76 MEN1 (0.55) MEN1MAPK1KMT2AGAACHRM1
SCHEMBL21773164 0.76 MEN1 (0.55) MEN1MAPK1KMT2AGAACHRM1
SCHEMBL21777609 0.76 MEN1 (0.55) MEN1MAPK1KMT2AGAACHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569646-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2005-09-07 EP disclosed
WO-2004054974-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2004-07-01 WO disclosed