SCHEMBL7464902

SCHEMBL7464902

CN1C2CCC1CC(Nc1ccccc1)C2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 3/20 0.54
CHRM5 P08912 3/20 0.54
HRH1 P35367 2/20 0.54
SIGMAR1 Q99720 2/20 0.54
HTR3E A5X5Y0 2/20 0.54
HTR3B O95264 2/20 0.54
CHRNA7 P36544 2/20 0.54
HTR3A P46098 2/20 0.54
HTR3D Q70Z44 2/20 0.54
HTR3C Q8WXA8 2/20 0.54
CHRNB2 P17787 1/20 0.54
CHRNB4 P30926 1/20 0.54
CHRNA3 P32297 1/20 0.54
CHRNA4 P43681 1/20 0.54
TMEM97 Q5BJF2 1/20 0.54
CHRM1 P11229 7/20 0.51
SLC6A2 P23975 6/20 0.51
SLC6A4 P31645 4/20 0.51
SLC6A3 Q01959 2/20 0.50
CARM1 Q86X55 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13850002 0.93 CHRM4 (0.59) CHRM4CHRM5HRH1SIGMAR1HTR3E
SCHEMBL2145704 0.93 CHRNA3 (0.63) CHRM4CHRM5HRH1SIGMAR1HTR3E
SCHEMBL12925024 0.91 CHRM4 (0.47) CHRM4CHRM5HRH1SIGMAR1HTR3E
SCHEMBL748392 0.80 HTR3E (0.50) CHRM4CHRM5HRH1SIGMAR1HTR3E
SCHEMBL748393 0.80 HTR3E (0.50) CHRM4CHRM5HRH1SIGMAR1HTR3E
SCHEMBL7457968 0.78 LMNA (0.49) HTR3ACHRM1SLC6A2SLC6A3CHRM3
SCHEMBL6153901 0.77 LTA4H (0.49) CHRM4CHRM5CHRM1OPRM1OPRD1
SCHEMBL6893103 0.77 HTR3E (0.54) CHRM4CHRM5HRH1SIGMAR1HTR3E
SCHEMBL6886547 0.77 HTR3E (0.54) CHRM4CHRM5HRH1SIGMAR1HTR3E
SCHEMBL14017444 0.76 HTR3A (0.60) CHRM4CHRM5HRH1SIGMAR1HTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242421-A1 4-[ARYL(8-AZABICYCLO[3.2.1] OCTAN-3-YL)] AMINOBENZOIC ACID DERIVATIVES Ortho-McNeil Pharmaceutical, Inc. (US) 2002-09-25 EP disclosed
US-6306876-B1 DRUGS WITH DIASTERIOMERS ORTHO-MCNEIL PHARMACEUTICAL, INC. 2001-10-23 US disclosed
WO-2001046191-A1 4-[ARYL(8-AZABICYCLO[3.2.1]OCTAN-3-YL)]AMINOBENZOIC ACID DERIVATIVES ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-06-28 WO disclosed