SCHEMBL6158768

SCHEMBL6158768

OCCC(Cn1ccnc1-c1ccccc1)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA3 P07451 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA13 Q8N1Q1 1/20 0.42
CA14 Q9ULX7 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
ESR1 P03372 1/20 0.41
PLAA Q9Y263 1/20 0.38
ALPG P10696 1/20 0.38
HTR1A P08908 1/20 0.35
HTR7 P34969 1/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
SLC6A2 P23975 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6160613 0.84 CA12 (0.41) CA12CA1CA2CA3CA4
SCHEMBL6166843 0.83 CA12 (0.41) CA12CA1CA2CA3CA4
SCHEMBL6160800 0.83 CA12 (0.41) CA12CA1CA2CA3CA4
SCHEMBL6159385 0.82 L3MBTL1 (0.37) HTR1AHTR7CYP3A4CYP2D6SLC6A2
Hydrochloric Acid SCHEMBL6159104 0.79 TACR2 (0.55) TACR2
SCHEMBL6160976 0.77 TSHR (0.46) HTR1AHTR7SLC6A2SLC6A3TSHR
SCHEMBL6160705 0.77 CYP11B1 (0.45) HTR1AHTR7CYP3A4CYP2D6SLC6A2
SCHEMBL6159965 0.77 TSHR (0.46) HTR1AHTR7SLC6A2SLC6A3TSHR
SCHEMBL6579685 0.75 HTT (0.34) TACR2HTT
SCHEMBL6579564 0.74 NPC1 (0.35) TACR2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0739891-B1 Substituted heterocycles ASTRAZENECA AB (SE) 2005-01-19 EP disclosed
US-6355695-B1 ANTIHISTAMINES; ASTHMA THERAPY ZENECA LIMITED (SE) 2002-03-12 US disclosed
US-6235757-B1 ANTIHISTAMINES ZENECA LIMITED (GB) 2001-05-22 US disclosed
US-6051580-A Substituted heterocycles ZENECA LIMITED 2000-04-18 US disclosed
US-5889024-A Substituted heterocycles ZENECA LIMITED (GB) 1999-03-30 US disclosed
EP-0739891-A2 Substituted heterocycles ZENECA LIMITED (GB) 1996-10-30 EP disclosed