SCHEMBL6161476

SCHEMBL6161476

COc1cc2ncnc(Nc3ccc(/C=C/C(=O)Nc4ccc(Cl)cc4)cc3)c2cc1OC

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDR P35968 15/20 0.69
FLT1 P17948 1/20 0.69
ABCG2 Q9UNQ0 1/20 0.65
EGFR P00533 3/20 0.64
HDAC3 O15379 6/20 0.64
HDAC1 Q13547 6/20 0.64
HDAC6 Q9UBN7 6/20 0.64
HDAC4 P56524 5/20 0.62
HDAC7 Q8WUI4 5/20 0.62
HDAC2 Q92769 5/20 0.62
HDAC10 Q969S8 5/20 0.62
HDAC11 Q96DB2 5/20 0.62
HDAC8 Q9BY41 5/20 0.62
HDAC9 Q9UKV0 5/20 0.62
HDAC5 Q9UQL6 5/20 0.62
AURKA O14965 1/20 0.59
AURKB Q96GD4 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6162791 1.00 KDR (0.69) KDRFLT1ABCG2EGFRHDAC3
SCHEMBL6162938 0.91 KDR (0.74) KDRABCG2EGFRHDAC3HDAC1
SCHEMBL6163496 0.91 KDR (0.70) KDRABCG2EGFRHDAC3HDAC1
SCHEMBL6166357 0.91 KDR (0.70) KDRABCG2EGFRHDAC3HDAC1
SCHEMBL6162947 0.91 KDR (0.74) KDRABCG2EGFRHDAC3HDAC1
SCHEMBL6164812 0.86 EGFR (0.66) KDRABCG2EGFRHDAC3HDAC1
SCHEMBL6164827 0.86 EGFR (0.66) KDRABCG2EGFRHDAC3HDAC1
SCHEMBL6161899 0.86 KDR (0.75) KDRFLT1ABCG2EGFRHDAC3
SCHEMBL6163629 0.86 KDR (0.75) KDRFLT1ABCG2EGFRHDAC3
SCHEMBL6165229 0.86 ABCG2 (0.64) KDRABCG2EGFRHDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218357-B1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2005-04-06 EP claimed