SCHEMBL6162947

SCHEMBL6162947

COc1cc2ncnc(Nc3ccc(C=CC(=O)Nc4ccccc4)cc3)c2cc1OC

nearest known ligand 0.74

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.74
AURKA O14965 2/20 0.68
AURKB Q96GD4 2/20 0.68
EGFR P00533 4/20 0.67
RET P07949 1/20 0.67
ABCG2 Q9UNQ0 4/20 0.66
LCK P06239 1/20 0.65
HDAC3 O15379 1/20 0.65
HDAC1 Q13547 1/20 0.65
HDAC6 Q9UBN7 1/20 0.65
ABCB1 P08183 3/20 0.64
SRC P12931 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6162938 1.00 KDR (0.74) KDRAURKAAURKBEGFRRET
SCHEMBL6166357 0.92 KDR (0.70) KDRAURKAAURKBEGFRRET
SCHEMBL6163496 0.92 KDR (0.70) KDRAURKAAURKBEGFRRET
SCHEMBL6161476 0.91 KDR (0.69) KDRAURKAAURKBEGFRABCG2
SCHEMBL6162791 0.91 KDR (0.69) KDRAURKAAURKBEGFRABCG2
SCHEMBL6161899 0.91 KDR (0.75) KDREGFRRETABCG2LCK
SCHEMBL6164827 0.91 EGFR (0.66) KDREGFRABCG2HDAC3HDAC1
SCHEMBL6163629 0.91 KDR (0.75) KDREGFRRETABCG2LCK
SCHEMBL6164812 0.91 EGFR (0.66) KDREGFRABCG2HDAC3HDAC1
SCHEMBL6165229 0.90 ABCG2 (0.64) KDRAURKAAURKBEGFRRET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218357-B1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2005-04-06 EP claimed