SCHEMBL6161611

SCHEMBL6161611

Cc1ccnc(C)c1C(=O)NN

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.54
KDM4E B2RXH2 4/20 0.43
ITGB1 P05556 1/20 0.42
ITGA4 P13612 1/20 0.42
MPO P05164 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2A6 P11509 1/20 0.41
CYP2C19 P33261 1/20 0.41
CCR5 P51681 1/20 0.40
SLC6A9 P48067 1/20 0.39
GAA P10253 5/20 0.38
ALDH1A1 P00352 5/20 0.38
MAPT P10636 2/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL351842 0.83 ITGB1 (0.40) P2RX7KDM4EITGB1ITGA4CYP1A2
SCHEMBL13687253 0.82 CCR5 (0.43) P2RX7KDM4EITGB1ITGA4CCR5
SCHEMBL161321 0.79 SIRT3 (0.46) P2RX7CCR5SLC6A9NOS3NOS2
SCHEMBL31606794 0.79 SIRT3 (0.46) P2RX7CCR5SLC6A9NOS3NOS2
SCHEMBL24571829 0.77 CYP1A2 (0.49) ITGB1ITGA4CYP1A2SLC6A9ALDH1A1
Hydrochloric Acid SCHEMBL5012214 0.77 NTRK1 (0.44) P2RX7CCR5SLC6A9NOS3NOS2
SCHEMBL9504646 0.77 CA1 (0.36) P2RX7ITGB1ITGA4CYP2A6CCR5
SCHEMBL29089331 0.77 NTRK1 (0.44) P2RX7CCR5SLC6A9NOS3NOS2
Hydrochloric Acid SCHEMBL5012204 0.77 NTRK1 (0.44) P2RX7CCR5SLC6A9NOS3NOS2
Iodide SCHEMBL27448063 0.77 NTRK1 (0.44) P2RX7CCR5SLC6A9NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1492784-A2 SUBSTITUTED 2,3-DIPHENYL PYRIDINES Merck & Co., Inc. (US) 2005-01-05 EP disclosed
WO-2003082191-A2 SUBSTITUTED 2,3-DIPHENYL PYRIDINES MERCK & CO., INC. (US) 2003-10-09 WO disclosed