SCHEMBL6161789

SCHEMBL6161789

C1=C(c2ccccc2)CCN(CCCCn2ccnn2)C1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.60
PARP1 P09874 2/20 0.49
DRD2 P14416 1/20 0.49
DRD4 P21917 1/20 0.49
DRD3 P35462 1/20 0.49
HTR1A P08908 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5846265 0.99 SIGMAR1 (0.59) SIGMAR1PARP1DRD2DRD4DRD3
SCHEMBL5846325 0.88 SIGMAR1 (0.48) SIGMAR1
SCHEMBL5846965 0.88 SIGMAR1 (0.62) SIGMAR1PARP1DRD2
SCHEMBL5846526 0.88 SIGMAR1 (0.62) SIGMAR1PARP1DRD2HTR1A
Hydrochloric Acid SCHEMBL5847835 0.86 SIGMAR1 (0.61) SIGMAR1PARP1DRD2HTR1A
Hydrochloric Acid SCHEMBL5846857 0.86 SIGMAR1 (0.47) SIGMAR1
Hydrochloric Acid SCHEMBL5847091 0.86 SIGMAR1 (0.61) SIGMAR1PARP1DRD2
SCHEMBL6159703 0.83 SIGMAR1 (0.62) SIGMAR1PARP1DRD2DRD4DRD3
Hydrochloric Acid SCHEMBL5846250 0.82 SIGMAR1 (0.60) SIGMAR1PARP1DRD2DRD4DRD3
SCHEMBL5846286 0.78 SIGMAR1 (0.61) SIGMAR1PARP1DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0721455-B9 TETRAHYDROPYRIDINE-(OR 4-HYDROXYPIPERIDINE)ALKYLAZOLES HAVING AN AFFINITY FOR SIGMA AND/OR 5HT1A RECEPTORS ESTEVE LABOR DR (ES) 2005-04-20 EP claimed
EP-0721455-B1 TETRAHYDROPYRIDINE-(OR 4-HYDROXYPIPERIDINE)ALKYLAZOLES HAVING AN AFFINITY FOR SIGMA AND/OR 5HT1A RECEPTORS ESTEVE LABOR DR (ES) 2002-12-11 EP claimed