SCHEMBL6161995

SCHEMBL6161995

COC(=O)C(N)(C(C)=O)c1cccc(N)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
KCNN4 O15554 1/20 0.42
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
DDX3X O00571 1/20 0.38
CYP3A4 P08684 1/20 0.37
PTGS1 P23219 3/20 0.37
F2 P00734 1/20 0.36
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
GAA P10253 2/20 0.35
PTPN1 P18031 1/20 0.35
PBRM1 Q86U86 1/20 0.34
NOS1 P29475 1/20 0.34
KDM4E B2RXH2 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3618566 0.84 KCNN4 (0.39) ALDH1A1KCNN4TSHRMAPK1DDX3X
SCHEMBL1068045 0.79 CNR1 (0.50) ALDH1A1KCNN4TSHRMAPK1DDX3X
SCHEMBL22165138 0.78 TSHR (0.52) ALDH1A1KCNN4TSHRMAPK1DDX3X
SCHEMBL7878585 0.76 TSHR (0.42) ALDH1A1TSHRMAPK1DDX3XCYP3A4
SCHEMBL3574723 0.76 TSHR (0.50) ALDH1A1KCNN4TSHRMAPK1DDX3X
SCHEMBL17978839 0.75 KCNN4 (0.50) ALDH1A1KCNN4TSHRMAPK1F2
SCHEMBL28918320 0.73 CA12 (0.41) ALDH1A1KCNN4TSHRCYP3A4MEN1
SCHEMBL19733460 0.73 TSHR (0.48) ALDH1A1TSHRMAPK1DDX3XCYP3A4
Acetic Acid Methyl Ester SCHEMBL28136526 0.72 ALDH1A1 (0.57) ALDH1A1TSHRDDX3XCYP3A4F2
SCHEMBL2237996 0.70 KCNN4 (0.37) ALDH1A1KCNN4TSHRMAPK1DDX3X

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1178969-B1 GASTRIN AND CHOLECYSTOKININ RECEPTOR LIGANDS BLACK JAMES FOUNDATION (GB) 2005-07-13 EP disclosed
US-6479531-B1 Gastrin and cholecystokinin receptor ligands JAMES BLACK FOUNDATION LIMITED (GB) 2002-11-12 US disclosed
EP-1178969-A1 GASTRIN AND CHOLECYSTOKININ RECEPTOR LIGANDS JAMES BLACK FOUNDATION LIMITED (GB) 2002-02-13 EP disclosed
WO-2000027823-A1 GASTRIN AND CHOLECYSTOKININ RECEPTOR LIGANDS JAMES BLACK FOUNDATION LIMITED (GB) 2000-05-18 WO disclosed