SCHEMBL6162253

SCHEMBL6162253

COc1ccc(-c2cc(C(=O)N3CCCC3CO)c3cccc(Cl)c3n2)c(F)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.46
HCRTR1 O43613 6/20 0.45
HCRTR2 O43614 6/20 0.45
RAB9A P51151 1/20 0.42
MAPT P10636 3/20 0.42
POLB P06746 1/20 0.41
ROCK2 O75116 1/20 0.40
HSP90AA1 P07900 1/20 0.40
NTRK1 P04629 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CPS1 P31327 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6161806 1.00 TRPV1 (0.46) TRPV1HCRTR1HCRTR2RAB9AMAPT
SCHEMBL6163596 1.00 TRPV1 (0.46) TRPV1HCRTR1HCRTR2RAB9AMAPT
SCHEMBL6163699 0.87 POLB (0.55) TRPV1HCRTR1HCRTR2RAB9AMAPT
SCHEMBL6163817 0.87 POLB (0.55) TRPV1HCRTR1HCRTR2RAB9AMAPT
SCHEMBL6165715 0.87 POLB (0.55) TRPV1HCRTR1HCRTR2RAB9AMAPT
SCHEMBL6161799 0.85 TRPV1 (0.44) TRPV1HCRTR1HCRTR2MAPTPOLB
SCHEMBL6163055 0.85 TRPV1 (0.44) TRPV1HCRTR1HCRTR2MAPTPOLB
SCHEMBL6162249 0.85 TRPV1 (0.44) TRPV1HCRTR1HCRTR2MAPTPOLB
SCHEMBL6167551 0.80 RAB9A (0.49) TRPV1HCRTR1HCRTR2RAB9ANTRK1
SCHEMBL6164221 0.80 TRPV1 (0.50) TRPV1HCRTR1HCRTR2MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1337523-B1 2,4-SUBSTITUTED PYRIDINE DERIVATIVES NEUROGEN CORP (US) 2005-10-19 EP claimed