SCHEMBL6162479

SCHEMBL6162479

N#CCCNc1ccc2ccccc2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.58
CYP1A2 P05177 3/20 0.58
CYP3A4 P08684 2/20 0.58
HSD17B10 Q99714 2/20 0.58
CYP2C19 P33261 2/20 0.58
HIF1A Q16665 2/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C9 P11712 1/20 0.58
HTT P42858 1/20 0.57
GAA P10253 3/20 0.53
THRB P10828 1/20 0.49
HPGD P15428 1/20 0.44
INSR P06213 1/20 0.44
IGF1R P08069 1/20 0.44
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
MAPT P10636 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
POLB P06746 1/20 0.41
NPC1 O15118 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11605746 0.82 CYP1A2 (0.75) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19
SCHEMBL11252585 0.79 HTT (0.61) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19
SCHEMBL11252528 0.78 GAA (0.70) ALDH1A1HTTGAATHRBHPGD
SCHEMBL4168758 0.77 ALDH1A1 (0.67) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19
SCHEMBL16366911 0.77 ALDH1A1 (0.51) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19
SCHEMBL141474 0.77 GAA (0.58) ALDH1A1HSD17B10HTTGAATHRB
SCHEMBL4341824 0.76 CYP1A2 (0.64) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19
SCHEMBL8808326 0.76 ALDH1A1 (0.64) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19
SCHEMBL11651781 0.76 ALDH1A1 (0.64) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19
SCHEMBL30447073 0.76 ALDH1A1 (0.64) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1210335-B1 AMINOCARBONYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES, METHOD FOR PRODUCING SAME AND THE USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA (DE) 2005-09-14 EP disclosed
US-6512000-B1 Aminocarbonyl- substituted benzimidazole derivatives for the treatment of diseases in which inhibition of tryptase is of therapeutic such as for treating an inflammatory or allergic disease BOEHRINGER INGELHEIM PHARMA KG (DE) 2003-01-28 US disclosed