SCHEMBL6163870

SCHEMBL6163870

CCON=Cc1cccc(-c2cc(=O)n(C)c3ccc(C(O)(c4ccc(Cl)cc4)c4cncn4C)cc23)c1

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FNTA P49354 9/20 0.72
FNTB P49356 9/20 0.72
CYP3A4 P08684 8/20 0.55
RORC P51449 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7672698 0.94 FNTA (0.69) FNTAFNTBCYP3A4RORC
SCHEMBL6163431 0.92 FNTA (0.75) FNTAFNTBCYP3A4RORC
SCHEMBL6163908 0.92 FNTA (0.68) FNTAFNTBCYP3A4RORC
SCHEMBL6161628 0.91 FNTA (0.73) FNTAFNTBCYP3A4RORC
SCHEMBL6165521 0.90 FNTA (0.79) FNTAFNTBCYP3A4RORC
SCHEMBL6165515 0.90 FNTA (0.79) FNTAFNTBCYP3A4RORC
SCHEMBL6165578 0.87 FNTA (0.82) FNTAFNTBCYP3A4RORC
SCHEMBL7044225 0.86 FNTA (0.81) FNTAFNTBCYP3A4RORC
SCHEMBL1683558 0.85 FNTA (0.79) FNTAFNTBCYP3A4RORC
SCHEMBL14588489 0.84 FNTA (0.71) FNTAFNTBCYP3A4RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1107962-B1 QUINOLIN-2-ONE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PROD INC (US) 2005-02-23 EP claimed
US-6495564-B1 SUCH AS 3-(6-((4-CHLORO-PHENYL)-HYDROXY-(3-METHYL-3H-IMIDAZOL-4-YL)-METHYL)-1-METHYL-2-OXO-1,2-DIHYDRO-QUINOLIN-4-YL)-BENZALDEHYDE O-METHYL-OXIME; INHIBITING ABNORMAL CELL GROWTH PFIZER INC. 2002-12-17 US claimed
EP-1107962-A1 QUINOLIN-2-ONE DERIVATIVES USEFUL AS ANTICANCER AGENTS Pfizer Products Inc. (US) 2001-06-20 EP claimed
WO-2000012498-A1 QUINOLIN-2-ONE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PRODUCTS INC. (US) 2000-03-09 WO claimed
EP-1107962-B1 QUINOLIN-2-ONE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PROD INC (US) 2005-02-23 EP disclosed
US-6495564-B1 SUCH AS 3-(6-((4-CHLORO-PHENYL)-HYDROXY-(3-METHYL-3H-IMIDAZOL-4-YL)-METHYL)-1-METHYL-2-OXO-1,2-DIHYDRO-QUINOLIN-4-YL)-BENZALDEHYDE O-METHYL-OXIME; INHIBITING ABNORMAL CELL GROWTH PFIZER INC. 2002-12-17 US disclosed
EP-1107962-A1 QUINOLIN-2-ONE DERIVATIVES USEFUL AS ANTICANCER AGENTS Pfizer Products Inc. (US) 2001-06-20 EP disclosed
WO-2000012498-A1 QUINOLIN-2-ONE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PRODUCTS INC. (US) 2000-03-09 WO disclosed