SCHEMBL6166236

SCHEMBL6166236

COc1c(N2CC[C@H](CC3(N)CC3)C2)c(F)cc2c(=O)c(C(=O)O)cn([C@@H]3C[C@H]3F)c12

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.67
CYP3A4 P08684 1/20 0.56
KDM4E B2RXH2 7/20 0.55
ALDH1A1 P00352 4/20 0.55
HPGD P15428 4/20 0.55
HSD17B10 Q99714 2/20 0.55
POLB P06746 2/20 0.55
TDP1 Q9NUW8 2/20 0.55
PRKD3 O94806 1/20 0.55
ALOX15 P16050 1/20 0.55
OPRM1 P35372 1/20 0.55
CLK2 P49760 1/20 0.55
CLK4 Q9HAZ1 1/20 0.55
TOP1 P11387 7/20 0.54
LMNA P02545 2/20 0.51
ATM Q13315 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6167085 1.00 KCNH2 (0.67) KCNH2CYP3A4KDM4EALDH1A1HPGD
SCHEMBL6168710 0.91 KCNH2 (0.57) KCNH2CYP3A4KDM4EALDH1A1HPGD
SCHEMBL27515036 0.91 KCNH2 (0.57) KCNH2CYP3A4KDM4EALDH1A1HPGD
SCHEMBL5546283 0.89 KCNH2 (0.73) KCNH2CYP3A4KDM4EALDH1A1HPGD
SCHEMBL6958823 0.87 CYP3A4 (0.74) KCNH2CYP3A4KDM4EALDH1A1HPGD
SCHEMBL6163513 0.85 CYP3A4 (0.50) KCNH2CYP3A4KDM4EALDH1A1HPGD
SCHEMBL30626289 0.85 KCNH2 (0.65) KCNH2CYP3A4KDM4EALDH1A1HPGD
SCHEMBL29080642 0.85 KCNH2 (0.65) KCNH2CYP3A4KDM4EALDH1A1HPGD
SCHEMBL5236833 0.84 CYP3A4 (0.65) KCNH2CYP3A4KDM4EALDH1A1HPGD
SCHEMBL5236827 0.84 CYP3A4 (0.65) KCNH2CYP3A4KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1134219-B1 CYCLOALKYL-SUBSTITUTED AMINOMETHYLPYRROLIDINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2005-06-15 EP disclosed
US-6573260-B1 Antibiotics DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2003-06-03 US disclosed