SCHEMBL6166716

SCHEMBL6166716

CCCN(CC(C)C)c1cc2c(cc1Cl)NC(=O)CC(c1cccc(-c3nc(CO)cs3)c1)=N2

nearest known ligand 0.44

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 5/20 0.44
CYP3A4 P08684 2/20 0.36
GRM3 Q14832 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6163335 0.89 GRM2 (0.47) GRM2CYP3A4GRM3
SCHEMBL6164544 0.89 GRM2 (0.47) GRM2CYP3A4GRM3
SCHEMBL6165782 0.89 GRM2 (0.49) GRM2CYP3A4GRM3
SCHEMBL6166445 0.86 GRM2 (0.51) GRM2CYP3A4GRM3
SCHEMBL6164053 0.85 GRM2 (0.49) GRM2CYP3A4GRM3
SCHEMBL6166940 0.82 CYP3A4 (0.42) GRM2CYP3A4GRM3
SCHEMBL6164871 0.79 GRM2 (0.49) GRM2CYP3A4GRM3
SCHEMBL6164581 0.79 GRM2 (0.52) GRM2CYP3A4GRM3
SCHEMBL5557071 0.78 GRM2 (0.57) GRM2CYP3A4
SCHEMBL6164951 0.78 GRM2 (0.44) GRM2CYP3A4GRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379511-B1 DIHYDRO-BENZO (b) (1, 4) DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II HOFFMANN LA ROCHE (CH) 2005-07-20 EP claimed