SCHEMBL6167070

SCHEMBL6167070

C=C(Cc1ccnc(-c2cc(OC)c(Cl)c(OC)c2)c1)N1CCC(=O)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 6/20 0.38
HCRTR2 O43614 6/20 0.38
WNK1 Q9H4A3 1/20 0.35
KDM1A O60341 1/20 0.34
HDAC1 Q13547 1/20 0.34
KDM4C Q9H3R0 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
EGFR P00533 1/20 0.33
TEC P42680 1/20 0.33
BTK Q06187 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE4B Q07343 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ERN1 O75460 1/20 0.33
KMO O15229 1/20 0.32
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6169530 0.91 HCRTR1 (0.39) HCRTR1HCRTR2KDM4EHSD17B10ABCB1
SCHEMBL6166854 0.86 HCRTR1 (0.36) HCRTR1HCRTR2PTGDR2PREPABCB1
Ethylene SCHEMBL4120382 0.83 PDE4D (0.43) HCRTR1HCRTR2WNK1HDAC1PDE4D
SCHEMBL4122248 0.83 PDE4D (0.45) HCRTR1HCRTR2WNK1HDAC1PDE4D
SCHEMBL4115040 0.74 RECQL (0.47) KDM1AHDAC1KDM4CERN1KMO
Ethylene SCHEMBL4115800 0.73 HCRTR1 (0.44) HCRTR1HCRTR2PDE4DKDM4EALDH1A1
SCHEMBL4114573 0.73 DYRK1A (0.39) HCRTR1HCRTR2KDM1AHDAC1KDM4C
SCHEMBL4117342 0.73 HCRTR1 (0.45) HCRTR1HCRTR2PDE4DKDM4EALDH1A1
SCHEMBL4114136 0.71 NPC1 (0.53) KDM4EALDH1A1NPC1
SCHEMBL27598696 0.70 PDE4D (0.43) HCRTR1HCRTR2PDE4DKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494670-A1 MEDICINE FOR TREATING CANCER Kowa Co., Ltd. (JP) 2005-01-12 EP disclosed
WO-2003086397-A1 MEDICINE FOR TREATING CANCER KOWA CO., LTD. (JP) 2003-10-23 WO disclosed