SCHEMBL61672

SCHEMBL61672

CCc1cccc(CC)c1-c1nc(C)c(COc2cc(C(C)C)ccc2C)c(C2=CCN(C(C)C(=O)O)CC2)n1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BCHE P06276 11/20 0.35
ACHE P22303 11/20 0.35
C5AR1 P21730 1/20 0.35
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HTT P42858 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
LMNA P02545 2/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
ALDH1A1 P00352 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
KEAP1 Q14145 1/20 0.31
NFE2L2 Q16236 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3509166 0.88 CCNT1 (0.36) BCHEACHEC5AR1CCNT1CDK9
SCHEMBL72861 0.88 C5AR1 (0.38) BCHEACHEC5AR1HTTSMN1; SMN2
SCHEMBL61126 0.86 BCHE (0.35) BCHEACHEC5AR1CCNT1CDK9
SCHEMBL73579 0.85 CCNT1 (0.36) BCHEACHEC5AR1CCNT1CDK9
SCHEMBL61151 0.85 PDK4 (0.40) BCHEACHE
SCHEMBL62101 0.81 C5AR1 (0.35) BCHEACHEC5AR1CCNT1CDK9
SCHEMBL62344 0.79 ACHE (0.43) BCHEACHEC5AR1HTTSMN1; SMN2
SCHEMBL3818877 0.78 ACHE (0.34) BCHEACHEC5AR1HTTSMN1; SMN2
SCHEMBL61659 0.77 C5AR1 (0.37) BCHEACHEC5AR1MEN1KMT2A
SCHEMBL13949214 0.76 BCHE (0.39) BCHEACHEMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129395-B2 4,5-disubstituted-2-aryl pyrimidines NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2012-03-06 US disclosed