SCHEMBL6167743

SCHEMBL6167743

C1CCOCC1.C1CCOCC1.O=C(O)CC(c1ccccc1)c1c[nH]c2cc(OCCCCNc3ccccn3)ccc12

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 20/20 0.48
ITGAV P06756 20/20 0.48
ITGB1 P05556 5/20 0.48
ITGB5 P18084 4/20 0.48
ITGB6 P18564 3/20 0.48
ITGA2B P08514 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dioxane SCHEMBL6167746 0.97 ITGB3 (0.49) ITGB3ITGAVITGB1ITGB5ITGB6
SCHEMBL3052806 0.94 ITGB3 (0.54) ITGB3ITGAVITGB1ITGB5ITGB6
SCHEMBL6162794 0.91 ITGB3 (0.57) ITGB3ITGAVITGB1ITGB5ITGB6
SCHEMBL3046153 0.91 ITGB3 (0.57) ITGB3ITGAVITGB1ITGB5ITGB6
Hydrochloric Acid SCHEMBL6696125 0.90 ITGB3 (0.56) ITGB3ITGAVITGB1ITGB5ITGB6
Trifluoroacetic Acid SCHEMBL6167633 0.89 ITGB3 (0.54) ITGB3ITGAVITGB1ITGB5ITGB6
SCHEMBL6697749 0.89 ITGB3 (0.53) ITGB3ITGAVITGB1ITGB5ITGB6
Trifluoroacetic Acid SCHEMBL6163896 0.87 ITGB3 (0.55) ITGB3ITGAVITGB1ITGB5ITGB6
SCHEMBL6165576 0.87 ITGB3 (0.52) ITGB3ITGAVITGB1ITGB5ITGB6
SCHEMBL3042341 0.87 ITGB3 (0.54) ITGB3ITGAVITGB1ITGB5ITGB6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1254133-B9 INDOL-3-YL DERIVATIVES AND THEIR USE AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2005-09-07 EP disclosed
EP-1254133-B1 INDOL-3-YL DERIVATIVES AND THEIR USE AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2005-04-20 EP disclosed
EP-1254133-A2 INDOL-3-YL DERIVATIVES MERCK PATENT GmbH (DE) 2002-11-06 EP disclosed
WO-2001058893-A2 INDOL-3-YL DERIVATIVES AND THEIR USE AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2001-08-16 WO disclosed