SCHEMBL6168890

SCHEMBL6168890

CC(C)C[C@H](OC(c1ccccc1)c1ccc(-c2ccc(CO)nc2O)cc1)C(=O)NCC#N

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSK P43235 16/20 0.47
CTSS P25774 10/20 0.47
CTSL P07711 9/20 0.43
CTSB P07858 5/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6168230 0.86 CTSK (0.49) CTSKCTSSCTSLCTSB
SCHEMBL6172109 0.85 CTSK (0.46) CTSKCTSSCTSLCTSB
SCHEMBL5513770 0.83 CTSK (0.55) CTSKCTSSCTSLCTSB
SCHEMBL5516794 0.81 CTSK (0.61) CTSKCTSSCTSLCTSB
SCHEMBL5518307 0.81 CTSK (0.61) CTSKCTSSCTSLCTSB
SCHEMBL5516415 0.81 CTSK (0.61) CTSKCTSSCTSLCTSB
SCHEMBL5514720 0.81 CTSK (0.61) CTSKCTSSCTSLCTSB
SCHEMBL5509563 0.81 CTSK (0.52) CTSKCTSSCTSLCTSB
SCHEMBL5513795 0.81 CTSK (0.59) CTSKCTSSCTSLCTSB
SCHEMBL5509541 0.80 CTSK (0.58) CTSKCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537074-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA INC. (CA) 2005-06-08 EP claimed
WO-2004022526-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA & CO. (CA) 2004-03-18 WO claimed