SCHEMBL6172878

SCHEMBL6172878

COc1ccc(-c2sc3ccccc3c2Cc2ccc(OCCN3CCCC3)cc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 9/20 0.66
ESR2 Q92731 9/20 0.66
F2 P00734 7/20 0.64
ITGA4 P13612 1/20 0.63
UBE2N P61088 1/20 0.62
LTA4H P09960 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6596926 0.95 ITGA4 (0.69) ESR1ESR2F2ITGA4LTA4H
SCHEMBL6596335 0.94 ITGA4 (0.68) ESR1ESR2F2ITGA4LTA4H
SCHEMBL6597629 0.91 F2 (0.67) ESR1ESR2F2ITGA4LTA4H
SCHEMBL7982501 0.91 F2 (0.67) ESR1ESR2F2ITGA4LTA4H
SCHEMBL6595837 0.91 F2 (0.76) ESR1ESR2F2ITGA4LTA4H
SCHEMBL7774025 0.91 F2 (0.65) ESR1ESR2F2ITGA4LTA4H
SCHEMBL7414082 0.90 F2 (0.64) ESR1ESR2F2ITGA4LTA4H
SCHEMBL7411720 0.90 F2 (0.75) ESR1ESR2F2ITGA4
SCHEMBL6171204 0.90 F2 (0.75) ESR1ESR2F2ITGA4
SCHEMBL6597039 0.90 F2 (0.64) ESR1ESR2F2ITGA4LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1027051-B1 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 2005-01-05 EP disclosed
US-6391901-B1 Thrombin inhibitors ELI LILLY AND COMPANY 2002-05-21 US disclosed
US-6288105-B1 COMPOUNDS SUCH AS (S)-2-(4-((2-AMINO-3-HYDROXY-1-OXOPROPYL)AMINO)PHENYL)-6-HYDRO XY-3-(3-METHOXY-4-(1-PYRROLIDINYLMETHYL)BENZYL)BENZO(B)THIOPHE NE ELI LILLY AND COMPANY 2001-09-11 US disclosed
US-6284756-B1 ANTICOAGULANT ELI LILLY AND COMPANY 2001-09-04 US disclosed
US-6271227-B1 ANTICOAGULANTS ELI LILLY AND COMPANY 2001-08-07 US disclosed