SCHEMBL6175152

SCHEMBL6175152

CC1(C)C(=O)N(c2ccc(OC(F)(F)F)cc2)C(=O)N1Cc1ncccc1C1CCCCC1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 16/20 0.44
GCGR P47871 2/20 0.37
NTRK1 P04629 1/20 0.36
CYP3A4 P08684 1/20 0.36
KCNH2 Q12809 1/20 0.36
EGLN2 Q96KS0 1/20 0.36
EGLN1 Q9GZT9 1/20 0.36
EGLN3 Q9H6Z9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6172608 0.83 IGF1R (0.46) IGF1REGLN2EGLN1EGLN3
SCHEMBL2940203 0.82 IGF1R (0.44) IGF1RGCGR
SCHEMBL2939387 0.81 IGF1R (0.56) IGF1RNTRK1
SCHEMBL6174193 0.77 IGF1R (0.48) IGF1R
SCHEMBL2939460 0.75 IGF1R (0.77) IGF1RGCGR
SCHEMBL2940116 0.74 IGF1R (0.69) IGF1R
SCHEMBL2939506 0.73 IGF1R (0.50) IGF1RGCGR
SCHEMBL2931702 0.73 IGF1R (0.60) IGF1RGCGR
SCHEMBL2937083 0.73 IGF1R (0.52) IGF1R
SCHEMBL2936903 0.72 IGF1R (0.72) IGF1RCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1599464-A2 NOVEL CYCLIC UREA DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL USE OF SAME AS KINASE INHIBITORS Aventis Pharma S.A. (FR) 2005-11-30 EP disclosed
WO-2004070050-A2 CYCLIC UREA DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL USE OF SAME AS KINASE INHIBITORS AVENTIS PHARMA S.A. (FR) 2004-08-19 WO disclosed