SCHEMBL6176597

SCHEMBL6176597

CC(C)(C)N1C(=O)C=C[C@]2(C)[C@H]3CC[C@]4(C)CCC[C@H]4[C@@H]3CC[C@@H]12

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MBOAT4 Q96T53 3/20 0.48
CYP19A1 P11511 3/20 0.47
AR P10275 5/20 0.47
KCNH2 Q12809 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9293075 0.89 AR (0.46) MBOAT4CYP19A1ARKCNH2
SCHEMBL9113552 0.84 AR (0.64) ARKCNH2
SCHEMBL14300609 0.84 AR (0.64) ARKCNH2
SCHEMBL9221841 0.84 AR (0.64) ARKCNH2
SCHEMBL7854363 0.80 AR (0.44) MBOAT4CYP19A1ARKCNH2
SCHEMBL15121576 0.74 AR (0.42) MBOAT4CYP19A1ARKCNH2
SCHEMBL9318018 0.74 CYP19A1 (0.44) CYP19A1
SCHEMBL29843057 0.74 CYP19A1 (0.44) CYP19A1
SCHEMBL4371413 0.73 AR (0.41) MBOAT4CYP19A1ARKCNH2
SCHEMBL9114762 0.73 AR (0.43) MBOAT4CYP19A1ARKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203770-B1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases UPJOHN CO (US) 2005-03-09 EP disclosed
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP disclosed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed