Betulinic Acid

Betulinic Acid

SCHEMBL61767

C=C(C)[C@@H]1CC[C@]2(C(=O)O)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 4/20 1.00
PTPN1 P18031 3/20 1.00
GPBAR1 Q8TDU6 3/20 1.00
ALB P02768 3/20 1.00
GLI1 P08151 2/20 1.00
USP2 O75604 2/20 1.00
LMNA P02545 2/20 1.00
HIF1A Q16665 2/20 1.00
AKR1B10 O60218 1/20 1.00
POLB P06746 1/20 1.00
AKR1B1 P15121 1/20 1.00
NT5E P21589 1/20 1.00
DPP4 P27487 1/20 1.00
SAE1 Q9UBE0 1/20 1.00
UBA2 Q9UBT2 1/20 1.00
EGLN2 Q96KS0 1/20 0.82
EGLN1 Q9GZT9 1/20 0.82
EGLN3 Q9H6Z9 1/20 0.82
P4HTM Q9NXG6 1/20 0.82
CES2 O00748 2/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Betulinic Acid SCHEMBL14112364 1.00 RORC (1.00) RORCPTPN1GPBAR1ALBGLI1
Betulinic Acid SCHEMBL13908717 1.00 RORC (1.00) RORCPTPN1GPBAR1ALBGLI1
Betulinic Acid SCHEMBL14112012 1.00 RORC (1.00) RORCPTPN1GPBAR1ALBGLI1
Betulinic Acid SCHEMBL7746410 1.00 RORC (1.00) RORCPTPN1GPBAR1ALBGLI1
Betulinic Acid SCHEMBL10214465 1.00 RORC (1.00) RORCPTPN1GPBAR1ALBGLI1
Betulinic Acid SCHEMBL9905925 1.00 RORC (1.00) RORCPTPN1GPBAR1ALBGLI1
Betulinic Acid SCHEMBL23132693 1.00 RORC (1.00) RORCPTPN1GPBAR1ALBGLI1
Betulinic Acid SCHEMBL13285621 1.00 RORC (1.00) RORCPTPN1GPBAR1ALBGLI1
Betulinic Acid SCHEMBL22251646 1.00 RORC (1.00) RORCPTPN1GPBAR1ALBGLI1
Betulinic Acid SCHEMBL21264235 1.00 RORC (1.00) RORCPTPN1GPBAR1ALBGLI1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 23282 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026105108-A2 AN ERGOTHIONEINE-CURCUMIN SYNERGISTIC ANTI-INFLAMMATORY AND ANTI-AGING COMPLEX COMPOSITION AND A PREPARATION METHOD THEREOF ZIRAOUI ANAS (EG) 2026-05-21 WO claimed
EP-3989943-B1 COMPOSITION COMPRISING AT LEAST ONE TRITERPENE AND/OR AT LEAST ONE TRITERPENOID AND/OR AT LEAST ONE OF THE GLYCOSYLATED FORMS THEREOF TILMAN (BE) 2026-05-20 EP claimed
EP-3841097-B1 2,6-BIS(((1H-BENZO[D]IMIDAZOL-2-YL)THIO)METHYL)PYRIDINE AND N2,N6-DIBENZYLPYRIDINE-2,6-DICARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS PHOSPHOINOSITIDE 3-KINASE (PI3K) INHIBITORS FOR TREATING CANCER BIOMEDICAL RES FOUNDATION OF THE ACADEMY OF ATHENS BRFAA (GR) 2026-05-20 EP claimed
CN-122056926-A Probiotic composition containing melatonin and application of composition in sleep 南京北极光生物科技有限公司 2026-05-19 CN claimed
CN-122060693-A Method for improving yield of betulinic acid synthesized by saccharomyces cerevisiae 江南大学 2026-05-19 CN claimed
US-20260130395-A1 Water Dispersible Botanical Compositions AQUILA BLACK LTD (AU) 2026-05-14 US claimed
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
EP-4694699-A2 COMPOSITIONS AND METHODS OF CONTROLLING MAMMALIAN SATIETY VitaKey Inc. (US) 2026-02-18 EP claimed
EP-4687999-A1 TROP2 CONJUGATED BIOLOGICAL MOLECULES, PHARMACEUTICAL COMPOSITIONS AND METHODS OBI Pharma, Inc. (TW) 2026-02-11 EP claimed
US-12544386-B2 Method and composition for treatment of skin diseases associated with accelerated corneodesmosomes degradation or weaker cell-cell adhesion ICHILOV TECH LTD (IL) 2026-02-10 US claimed
WO-1998043936-A2 IMPROVED METHODS OF MANUFACTURING BETULINIC ACID THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 1998-10-08 WO claimed
US-5804575-A Methods of manufacturing betulinic acid THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 1998-09-08 US claimed
CN-1177480-A Preparation absorbed through skin, containing woluoke kinds of medicine HU YOUPU (CN) 1998-04-01 CN claimed
EP-0814795-A2 USE OF BETULINIC ACID AND ITS DERIVATIVES FOR INHIBITING MALIGNANT MELANOMA GROWTH AND A METHOD OF MONITORING THIS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 1998-01-07 EP claimed
CN-1163643-A Method for production of creped hygienic cellulose paper PROCTER & GAMBLE (US) 1997-10-29 CN claimed
US-5658947-A TOPICALLY APPLYING BETULINIC ACID OR DERIVATIVE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 1997-08-19 US claimed
WO-1996029068-A2 USE OF BETULINIC ACID AND ITS DERIVATIVES FOR INHIBITING MALIGNANT MELANOMA GROWTH AND A METHOD OF MONITORING THIS BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 1996-09-26 WO claimed
EP-0717983-A1 Cosmetic compositions containing betulinic acid UNILEVER PLC (GB) 1996-06-26 EP claimed
US-5529769-A REDUCING SIGNS OF AGING CHESEBROUGH-POND'S USA CO., DIVISION OF CONOPCO, INC. (US) 1996-06-25 US claimed
CN-1045784-A Speiss in the camptothecine production process is handled GUANGXI HECHI DISTRICT TECHNOL (CN) 1990-10-03 CN claimed