SCHEMBL6177634

SCHEMBL6177634

CCn1nc(-c2ccc(F)cc2)c(-c2ccncc2)c1NC(=O)Cc1ccccn1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 13/20 0.49
RAB9A P51151 1/20 0.41
EGFR P00533 1/20 0.40
RAF1 P04049 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
GSK3B P49841 1/20 0.40
RIPK3 Q9Y572 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
SRC P12931 1/20 0.40
BRAF P15056 1/20 0.40
KDR P35968 1/20 0.40
PTGS2 P35354 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4348734 0.88 MAPK14 (0.63) MAPK14EGFRRAF1ADORA3ADORA2A
SCHEMBL7134709 0.88 MAPK14 (0.56) MAPK14RAB9AEGFRRAF1ADORA3
SCHEMBL6176484 0.86 MAPK14 (0.53) MAPK14RAB9AEGFRRAF1ADORA3
SCHEMBL4338046 0.82 MAPK14 (0.65) MAPK14EGFRRAF1ADORA3ADORA2A
SCHEMBL6175447 0.81 MAPK14 (0.45) MAPK14EGFRRAF1ADORA3ADORA2A
SCHEMBL6029490 0.80 SMN1; SMN2 (0.47) MAPK14RAB9A
SCHEMBL4348737 0.79 MAPK14 (0.49) MAPK14EGFRRAF1ADORA3ADORA2A
SCHEMBL6176488 0.79 MAPK14 (0.45) MAPK14EGFRRAF1ADORA3ADORA2A
SCHEMBL6179804 0.78 MAPK14 (0.63) MAPK14EGFRRAF1ADORA3ADORA2A
SCHEMBL6029308 0.77 TACR1 (0.41) MAPK14EGFRRAF1ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1142890-B1 AMINOPYRAZOLE DERIVATIVES TEIKOKU HORMONE MFG CO LTD (JP) 2005-08-03 EP disclosed
US-6511997-B1 For treatment of a disease associated with tumor necrosis factor alpha, interleukin 1, interleukin 6 or cyclooxygenase II; such as irritable bowel disease TEIKOKU HORMONE MFG. CO., LTD. (JP) 2003-01-28 US disclosed
EP-1142890-A1 AMINOPYRAZOLE DERIVATIVES TEIKOKU HORMONE MFG. CO., LTD. (JP) 2001-10-10 EP disclosed