SCHEMBL6179865

SCHEMBL6179865

Cc1ncc(C=C(Cc2cccs2)C(=O)O)n1Cc1ccc(Cl)cc1Cl

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 4/20 0.61
ABCC3 O15438 1/20 0.51
ABCC2 Q92887 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6179859 1.00 AGTR1 (0.61) AGTR1ABCC3ABCC2
SCHEMBL6181485 0.86
SCHEMBL6181480 0.86
SCHEMBL6181764 0.83 AGTR1 (0.51) AGTR1
SCHEMBL6181752 0.83 AGTR1 (0.51) AGTR1
SCHEMBL6972699 0.80 AGTR1 (0.72) AGTR1
SCHEMBL6972690 0.80 AGTR1 (0.72) AGTR1
SCHEMBL6972507 0.79 AGTR1 (0.84) AGTR1
SCHEMBL6972501 0.79 AGTR1 (0.84) AGTR1
SCHEMBL6642074 0.78 AGTR1 (0.81) AGTR1ABCC3ABCC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000932-B9 AROMATIC RING DERIVATIVES FUJISAWA PHARMACEUTICAL CO (JP) 2005-12-28 EP disclosed
EP-1000932-B1 AROMATIC RING DERIVATIVES FUJISAWA PHARMACEUTICAL CO (JP) 2004-09-15 EP disclosed
US-6242474-B1 SULFONYLCARBAMOYLALKYLIMIDAZOLE DERIVATIVES; ANTIDIABETIC AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-06-05 US disclosed
EP-1000932-A1 AROMATIC RING DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-05-17 EP disclosed