SCHEMBL6180381

SCHEMBL6180381

CCN(CC)CCN1C(=O)C(O)(c2ccc3ccccc3c2)c2c1cc(C(=O)N(C)C)cc2C(F)(F)F

nearest known ligand 0.83

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 16/20 0.83
POLB P06746 1/20 0.33
PDK2 Q15119 1/20 0.32
SCN9A Q15858 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6176838 0.91 GHSR (1.00) GHSRPOLBKMT2A
SCHEMBL6179679 0.90 GHSR (0.83) GHSRPOLB
SCHEMBL6176424 0.89 GHSR (0.81) GHSRKMT2A
SCHEMBL7855537 0.86 GHSR (0.77) GHSRKMT2A
SCHEMBL6176208 0.86 GHSR (0.77) GHSRPOLBSCN9AKMT2A
SCHEMBL6180076 0.86 GHSR (0.76) GHSRPOLBSCN9A
SCHEMBL6179027 0.85 GHSR (0.75) GHSR
SCHEMBL6176866 0.84 GHSR (0.73) GHSR
SCHEMBL6180879 0.84 GHSR (0.73) GHSRPOLBSCN9AKMT2A
SCHEMBL6180416 0.84 GHSR (0.82) GHSRSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1105376-B1 OXINDOLE DERIVATIVES AS GROWTH HORMONE RELEASERS SUMITOMO PHARMA (JP) 2005-02-09 EP disclosed
US-6576656-B1 Such as 1-(2-diethylaminoethyl)-4-trifluoromethyl-6-carbamoyl-3-hydroxy-3-(2 -chlorophenyl)oxindole; growth hormone releaser SUMITOMO PHARMACEUTICALS CO., LTD. (JP) 2003-06-10 US disclosed