Fluoroacetate

Fluoroacetate

SCHEMBL6182223

N=C(N)c1cccc(C2=C(C(=O)Nc3ccc(-c4ccccn4)cc3)CCC2)c1.O=C(O)CF

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
F10 P00742 9/20 0.46
PRSS1 P07477 9/20 0.46
PRSS2 P07478 8/20 0.46
PRSS3 P35030 8/20 0.46
F2 P00734 7/20 0.46
TRPV1 Q8NER1 2/20 0.44
DHODH Q02127 1/20 0.42
CNR1 P21554 1/20 0.42
PLAU P00749 1/20 0.41
PLAT P00750 1/20 0.41
CREBBP Q92793 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6164497 0.92 F10 (0.54) F10PRSS1PRSS2PRSS3F2
Fluoroacetate SCHEMBL6182231 0.84 TRPV1 (0.41) TRPV1DHODHCNR1CREBBP
SCHEMBL6171566 0.78 GRM4 (0.54) TRPV1DHODHCNR1CREBBP
Trifluoroacetic Acid SCHEMBL6164502 0.77 TRPV1 (0.44) F10PRSS1PRSS2PRSS3F2
SCHEMBL7494748 0.76 F10 (0.73) F10PRSS1PRSS2PRSS3F2
Trifluoroacetic Acid SCHEMBL6203384 0.75 F10 (0.76) F10PRSS1PRSS2PRSS3F2
Trifluoroacetic Acid SCHEMBL6238656 0.73 F10 (0.51) F10PRSS1PRSS2PRSS3F2
SCHEMBL6840558 0.72 F10 (0.58) F10PRSS1F2
Acetic Acid SCHEMBL6839721 0.71 F10 (0.57) F10PRSS1F2
SCHEMBL18573213 0.68 TRPV1 (0.71) TRPV1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1254136-A4 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD (KR) 2005-06-01 EP claimed
EP-1254136-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG Chem Investment, Ltd. (KR) 2002-11-06 EP claimed
WO-2001055146-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD. (KR) 2001-08-02 WO claimed