Fluoroacetate

Fluoroacetate

SCHEMBL6182231

NN=Cc1cccc(C2=C(C(=O)Nc3ccc(-c4ccccn4)cc3)CCC2)c1.O=C(O)CF

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.41
DHODH Q02127 1/20 0.41
PORCN Q9H237 1/20 0.41
CNR1 P21554 1/20 0.39
CREBBP Q92793 1/20 0.38
SMO Q99835 2/20 0.37
CYP2C9 P11712 1/20 0.36
NR4A2 P43354 1/20 0.36
CHRNA7 P36544 1/20 0.36
PTPN2 P17706 1/20 0.36
PTPN1 P18031 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6164502 0.92 TRPV1 (0.44) TRPV1DHODHPORCNCNR1CREBBP
Fluoroacetate SCHEMBL6182223 0.84 F10 (0.46) TRPV1DHODHCNR1CREBBP
Trifluoroacetic Acid SCHEMBL6164497 0.77 F10 (0.54) TRPV1
SCHEMBL6171566 0.77 GRM4 (0.54) TRPV1DHODHCNR1CREBBP
Trifluoroacetic Acid SCHEMBL7101440 0.76 F10 (0.54)
Trifluoroacetic Acid SCHEMBL6238659 0.75 DHODH (0.39) DHODHNR4A2
Fluoroacetate SCHEMBL6182226 0.74 HDAC3 (0.35) DHODH
Trifluoroacetic Acid SCHEMBL6161749 0.70 F10 (0.47)
SCHEMBL18573213 0.64 TRPV1 (0.71) TRPV1CNR1PTPN2PTPN1
SCHEMBL7950222 0.64 CA12 (0.59) CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1254136-A4 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD (KR) 2005-06-01 EP claimed
EP-1254136-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG Chem Investment, Ltd. (KR) 2002-11-06 EP claimed
WO-2001055146-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD. (KR) 2001-08-02 WO claimed