Fluoroacetate

Fluoroacetate

SCHEMBL6182226

NN=Cc1cccc(C2=C(C(N)=O)CCC2c2ccc(-c3ccccn3)cc2)c1.O=C(O)CF

nearest known ligand 0.35

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 2/20 0.33
SYK P43405 3/20 0.33
DGAT1 O75907 1/20 0.33
KDM1A O60341 1/20 0.32
SIRT1 Q96EB6 2/20 0.32
SIRT2 Q8IXJ6 1/20 0.32
SIRT3 Q9NTG7 1/20 0.32
FFAR1 O14842 1/20 0.32
TLR4 O00206 1/20 0.32
TLR2 O60603 1/20 0.32
PARP1 P09874 1/20 0.31
DHODH Q02127 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
AKT1 P31749 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6171571 0.77 GRM5 (0.43) KDM1APARP1DHODHPARP2
Trifluoroacetic Acid SCHEMBL6164502 0.67 TRPV1 (0.44) DHODHF2F10
SCHEMBL3814048 0.63 CA12 (0.59) HDAC3HDAC1HDAC2CA12CA1
SCHEMBL3814046 0.63 CA12 (0.59) HDAC3HDAC1HDAC2CA12CA1
SCHEMBL7950222 0.63 CA12 (0.59) HDAC3HDAC1HDAC2CA12CA1
Hydrochloric Acid SCHEMBL9769062 0.62 CA12 (0.58) HDAC3HDAC1HDAC2CA12CA1
SCHEMBL6168451 0.61 CYP11B2 (0.43) KDM1A
Cyanide SCHEMBL22130168 0.60 CA12 (0.56) HDAC3HDAC1HDAC2CA12CA1
SCHEMBL25398509 0.59 TLR4 (0.55) CA12CA1CA2CA9KDM1A
SCHEMBL30036208 0.59 CHEK2 (0.57) SYKKDM1APARP1DHODHCHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1254136-A4 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD (KR) 2005-06-01 EP claimed
EP-1254136-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG Chem Investment, Ltd. (KR) 2002-11-06 EP claimed
WO-2001055146-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD. (KR) 2001-08-02 WO claimed