SCHEMBL6182397

SCHEMBL6182397

Cn1cnc(COc2ccc(-c3cc(-c4c[nH]c(-n5ccc(-c6ccccn6)c5)c4)ccn3)cc2)c1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMO Q99835 3/20 0.40
MAPK14 Q16539 2/20 0.40
TGFBR1 P36897 7/20 0.38
CYP2C9 P11712 3/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP19A1 P11511 1/20 0.36
CYP2C19 P33261 1/20 0.36
ACVR1B P36896 1/20 0.35
GRM5 P41594 1/20 0.35
KCNH2 Q12809 1/20 0.34
FFAR1 O14842 3/20 0.33
COMT P21964 1/20 0.33
CYP3A4 P08684 1/20 0.33
KDM2B Q8NHM5 1/20 0.33
PHF8 Q9UPP1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6182965 0.78 TGFBR1 (0.46) SMOMAPK14TGFBR1CYP2C9CYP1A2
SCHEMBL6327640 0.72 TGFBR1 (0.40) SMOMAPK14TGFBR1CYP2C9ACVR1B
SCHEMBL5907466 0.70 TGFBR1 (0.41) MAPK14TGFBR1
SCHEMBL5790048 0.66 TGFBR1 (0.38) SMOMAPK14TGFBR1
SCHEMBL5956566 0.65 TGFBR1 (0.52) MAPK14TGFBR1
SCHEMBL6181800 0.62 TGFBR1 (0.46) TGFBR1CYP2C9CYP1A2CYP2D6CYP19A1
SCHEMBL29348729 0.61 SMN1; SMN2 (0.48) CYP2C9CYP19A1CYP2C19KCNH2
SCHEMBL6180723 0.61 TGFBR1 (0.49) TGFBR1CYP2C9CYP1A2CYP2D6CYP19A1
SCHEMBL29348730 0.60 APP (0.47) CYP2C9CYP2C19
SCHEMBL12339143 0.60 TGFBR1 (0.63) TGFBR1CYP2C9CYP1A2CYP2D6CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355903-B1 PYRAZOLE DERIVATIVES AGAINST TGF OVEREXPRESSION SMITHKLINE BEECHAM CORP (US) 2005-03-16 EP claimed