SCHEMBL6184426

SCHEMBL6184426

Cc1ccc(CCNCc2ccc(Oc3ccc(C(N)=O)nc3)c(F)c2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 7/20 0.61
OPRD1 P41143 6/20 0.61
OPRK1 P41145 6/20 0.61
ROCK1 Q13464 2/20 0.43
GRIN2D O15399 1/20 0.43
GRIN3B O60391 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A3 Q01959 1/20 0.43
GRIN1 Q05586 1/20 0.43
KCNH2 Q12809 1/20 0.43
GRIN2A Q12879 1/20 0.43
GRIN2B Q13224 1/20 0.43
GRIN2C Q14957 1/20 0.43
GRIN3A Q8TCU5 1/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HTT P42858 1/20 0.42
PPARD Q03181 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3696666 0.92 OPRM1 (0.63) OPRM1OPRD1OPRK1ROCK1GRIN2D
SCHEMBL3700784 0.91 OPRM1 (0.60) OPRM1OPRD1OPRK1ROCK1GRIN2D
SCHEMBL3695213 0.87 OPRM1 (0.57) OPRM1OPRD1OPRK1ROCK1GRIN2D
SCHEMBL3696696 0.86 OPRM1 (0.61) OPRM1OPRD1OPRK1ROCK1GRIN2D
SCHEMBL3692278 0.86 OPRM1 (0.61) OPRM1OPRD1OPRK1ROCK1GRIN2D
SCHEMBL3695517 0.85 OPRM1 (0.52) OPRM1OPRD1OPRK1PPARDCARM1
SCHEMBL3689306 0.85 OPRM1 (0.52) OPRM1OPRD1OPRK1PPARDCARM1
SCHEMBL13773070 0.85 OPRM1 (0.52) OPRM1OPRD1OPRK1CYP3A4CYP2D6
SCHEMBL3698265 0.84 OPRM1 (0.50) OPRM1OPRD1OPRK1PPARDCARM1
SCHEMBL3698271 0.84 OPRM1 (0.50) OPRM1OPRD1OPRK1PPARDCARM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562595-A1 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2005-08-17 EP disclosed
WO-2004026305-A1 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONIST ELI LILLY AND COMPANY (US) 2004-04-01 WO disclosed