SCHEMBL6184715

SCHEMBL6184715

CN(Cc1cccc(-c2ccc(/C=C3\SC(=O)NC3=O)cc2)c1)c1ccccn1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARG P37231 3/20 0.52
PTPN1 P18031 4/20 0.50
HPGD P15428 6/20 0.49
POLB P06746 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
GSK3B P49841 1/20 0.46
MAOA P21397 1/20 0.45
MAOB P27338 1/20 0.45
PIM1 P11309 2/20 0.43
PIM2 Q9P1W9 2/20 0.43
PIM3 Q86V86 1/20 0.43
NAT1 P18440 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6184718 1.00 PPARG (0.52) PPARGPTPN1HPGDPOLBMEN1
SCHEMBL6186299 0.81 HIF1A (0.42) PPARGPOLBKMT2A
SCHEMBL5397253 0.79 MEN1 (0.53) PTPN1HPGDPOLBMEN1KMT2A
SCHEMBL5397249 0.79 MEN1 (0.53) PTPN1HPGDPOLBMEN1KMT2A
SCHEMBL6185163 0.77 HSD17B2 (0.51) PTPN1HPGDPOLBMEN1KMT2A
SCHEMBL6185166 0.77 HSD17B2 (0.51) PTPN1HPGDPOLBMEN1KMT2A
SCHEMBL6184071 0.76 MEN1 (0.47) PTPN1HPGDPOLBMEN1KMT2A
SCHEMBL6184070 0.76 MEN1 (0.47) PTPN1HPGDPOLBMEN1KMT2A
SCHEMBL6182018 0.76 HPGD (0.54) PTPN1HPGDKMT2ANAT1
SCHEMBL6182023 0.76 HPGD (0.54) PTPN1HPGDKMT2ANAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1309575-B1 BIPHENYL DERIVATIVES AND THEIR USE AS PPAR-GAMMA RECEPTOR ACTIVATORS GALDERMA RES & DEV (FR) 2005-06-08 EP disclosed
EP-1309575-A1 BIPHENYL DERIVATIVES AND THEIR USE AS PPAR-GAMMA RECEPTOR ACTIVATORS Galderma Research & Development (FR) 2003-05-14 EP disclosed
WO-2002012210-A9 BIPHENYL DERIVATIVES AND THEIR USE AS PPAR-GAMMA RECEPTOR ACTIVATORS GALDERMA RES & DEV (FR) 2002-04-18 WO disclosed
WO-2002012210-A1 BIPHENYL DERIVATIVES AND THEIR USE AS PPAR-GAMMA RECEPTOR ACTIVATORS GALDERMA RESEARCH & DEVELOPMENT (FR) 2002-02-14 WO disclosed