SCHEMBL6185585

SCHEMBL6185585

COc1cccc(OC2CN(CC(C)O)CCN2)c1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
GRIN2B Q13224 3/20 0.40
GRIN1 Q05586 1/20 0.40
SLC6A2 P23975 3/20 0.40
MAPT P10636 1/20 0.39
GAA P10253 1/20 0.39
KDM4E B2RXH2 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6184734 0.88 GRIN1 (0.40) L3MBTL1GRIN2BGRIN1SLC6A2MAPT
SCHEMBL2331866 0.81 CHRM2 (0.36) MAPT
SCHEMBL8349073 0.81 USP2 (0.41) MAPT
Hydrochloric Acid SCHEMBL11619919 0.75 KMT2A (0.42) MAPTKDM4E
SCHEMBL6186053 0.75 CYP3A4 (0.41)
SCHEMBL5745430 0.75 CYP3A4 (0.41)
SCHEMBL6185503 0.75 L3MBTL1 (0.39) L3MBTL1MAPTKDM4E
Hydrochloric Acid SCHEMBL11620280 0.74 SMN1; SMN2 (0.36)
SCHEMBL27682123 0.74 SMN1; SMN2 (0.35)
SCHEMBL6185575 0.73 NPC1 (0.40) TP53L3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567525-A2 SUBSTITUTED PIPERAZINE COMPOUNDS AND THEIR USE AS FATTY ACID OXIDATION INHIBITORS CV THERAPEUTICS, INC. (US) 2005-08-31 EP disclosed
WO-2004052887-A2 SUBSTITUTED PIPERAZINE COMPOUNDS AND THEIR USE AS FATTY ACID OXIDATION INHIBITORS CV THERAPEUTICS, INC. (US) 2004-06-24 WO disclosed