SCHEMBL6186145

SCHEMBL6186145

N#Cc1ccc(C(F)(F)F)nc1OCC[C@H](N)C(O)c1ccno1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.59
NOS2 P35228 2/20 0.59
CYP3A4 P08684 1/20 0.33
AAK1 Q2M2I8 1/20 0.33
MBOAT4 Q96T53 2/20 0.32
GPR119 Q8TDV5 1/20 0.32
TRPV1 Q8NER1 1/20 0.31
SCN9A Q15858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6286190 0.84 SLC6A4 (0.62) SLC6A4NOS2CYP3A4AAK1MBOAT4
SCHEMBL6280985 0.76 SLC6A4 (0.49) SLC6A4NOS2CYP3A4AAK1MBOAT4
SCHEMBL2532315 0.75 SLC6A4 (0.49) SLC6A4NOS2CYP3A4AAK1GPR119
SCHEMBL6050236 0.74 SLC6A4 (1.00) SLC6A4NOS2CYP3A4AAK1GPR119
SCHEMBL6892410 0.74 SLC6A4 (1.00) SLC6A4NOS2CYP3A4AAK1GPR119
SCHEMBL6186136 0.73 SLC6A4 (0.71) SLC6A4NOS2CYP3A4AAK1GPR119
SCHEMBL6050141 0.73 SLC6A4 (0.88) SLC6A4NOS2CYP3A4AAK1GPR119
SCHEMBL6285580 0.71 SLC6A4 (0.45) SLC6A4NOS2CYP3A4AAK1MBOAT4
SCHEMBL2528648 0.71 SLC6A4 (0.46) SLC6A4NOS2MBOAT4GPR119TRPV1
SCHEMBL6050379 0.70 SLC6A4 (0.76) SLC6A4NOS2GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1572655-A2 NOVEL ARYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2005-09-14 EP claimed
WO-2002090332-A2 NOVEL AEYLHETEROALKYLAMINΕ DERIVATIVES ASTRAZENECA AB (SE) 2002-11-14 WO claimed
EP-1572655-A2 NOVEL ARYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2005-09-14 EP disclosed
WO-2002090332-A2 NOVEL AEYLHETEROALKYLAMINΕ DERIVATIVES ASTRAZENECA AB (SE) 2002-11-14 WO disclosed