SCHEMBL6186910

SCHEMBL6186910

O=C(O)C=CNC(=O)Cc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
EPHX2 P34913 2/20 0.52
GAA P10253 2/20 0.50
HPGD P15428 1/20 0.50
TRPV1 Q8NER1 1/20 0.47
ALDH1A1 P00352 4/20 0.47
CNR2 P34972 4/20 0.47
LMNA P02545 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
AKR1B1 P15121 1/20 0.47
TAAR1 Q96RJ0 2/20 0.46
ATM Q13315 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21333228 1.00 MEN1 (0.55) MEN1KMT2AHDAC8HDAC6EPHX2
SCHEMBL27370508 0.83 ALDH1A1 (0.49) MEN1KMT2AHDAC8HDAC6EPHX2
SCHEMBL11153839 0.81 MEN1 (0.55) MEN1KMT2AHDAC8HDAC6EPHX2
SCHEMBL11153843 0.81 MEN1 (0.55) MEN1KMT2AHDAC8HDAC6EPHX2
SCHEMBL11153841 0.81 MEN1 (0.55) MEN1KMT2AHDAC8HDAC6EPHX2
SCHEMBL27865872 0.80 CNR2 (0.59) MEN1KMT2AHDAC8HDAC6EPHX2
SCHEMBL10585859 0.79 MEN1 (0.57) MEN1KMT2AHDAC8HDAC6EPHX2
SCHEMBL6253478 0.79 MEN1 (0.57) MEN1KMT2AHDAC8HDAC6EPHX2
SCHEMBL30866449 0.79 MAPT (0.57) MEN1KMT2AHDAC8HDAC6HPGD
SCHEMBL2750185 0.79 MEN1 (0.61) MEN1KMT2AHDAC8HDAC6EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532128-A1 INHIBITORS OF HCV NS5B POLYMERASE Pharmacia & Upjohn Company LLC (US) 2005-05-25 EP disclosed
WO-2004002977-A1 INHIBITORS OF HCV NS5B POLYMERASE PHARMACIA & UPJOHN COMPANY LLC (US) 2004-01-08 WO disclosed