SCHEMBL6188415

SCHEMBL6188415

CC(CNC(=O)CC1NC(=O)NC1=O)c1ccc(Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.52
KDM4E B2RXH2 7/20 0.52
GAA P10253 5/20 0.52
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
CASP1 P29466 1/20 0.43
HSD17B10 Q99714 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
ALOX15 P16050 1/20 0.42
LMNA P02545 1/20 0.41
POLB P06746 3/20 0.40
MAPT P10636 3/20 0.40
OPRM1 P35372 1/20 0.40
NTSR1 P30989 1/20 0.40
HTT P42858 1/20 0.40
P2RX7 Q99572 1/20 0.39
ADAMTS5 Q9UNA0 2/20 0.39
MMP2 P08253 1/20 0.39
ADAM17 P78536 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2875815 0.86 ALDH1A1 (0.48) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL2872252 0.85 ALDH1A1 (0.47) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL2873664 0.83 ALDH1A1 (0.46) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL2871365 0.83 GAA (0.43) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL2874347 0.82 ALDH1A1 (0.61) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL2872368 0.81 ALDH1A1 (0.47) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL2872321 0.80 ALDH1A1 (0.45) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL2874185 0.79 MAPT (0.46) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL2865278 0.79 ALDH1A1 (0.47) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL2870693 0.79 ALDH1A1 (0.44) ALDH1A1KDM4EGAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542977-A1 2,5-DIOXOIMIDAZOLIDIN-4-YL ACETAMIDES AND ANALOGUES AS INHIBITORS OF METALLOPROTEINASE MMP12. AstraZeneca AB (SE) 2005-06-22 EP claimed
WO-2004020415-A1 2,5-DIOXOIMIDAZOLIDIN-4-YL ACETAMIDES AND ANALOGUES AS INHIBITORS OF METALLOPROTEINASE MMP12. ASTRAZENECA AB (SE) 2004-03-11 WO claimed
EP-1542977-A1 2,5-DIOXOIMIDAZOLIDIN-4-YL ACETAMIDES AND ANALOGUES AS INHIBITORS OF METALLOPROTEINASE MMP12. AstraZeneca AB (SE) 2005-06-22 EP disclosed
WO-2004020415-A1 2,5-DIOXOIMIDAZOLIDIN-4-YL ACETAMIDES AND ANALOGUES AS INHIBITORS OF METALLOPROTEINASE MMP12. ASTRAZENECA AB (SE) 2004-03-11 WO disclosed