SCHEMBL6196178

SCHEMBL6196178

O=c1nc(-c2ccc(F)c(F)c2)cc[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.46
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C8 P10632 1/20 0.45
TGFBR1 P36897 1/20 0.45
MAOB P27338 2/20 0.42
TRPV3 Q8NET8 1/20 0.42
ALDH1A1 P00352 2/20 0.40
GAA P10253 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
NOTUM Q6P988 1/20 0.40
RAB9A P51151 3/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
TYMP P19971 1/20 0.38
GPR84 Q9NQS5 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPK1 P28482 1/20 0.37
PSMD14 O00487 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4903170 0.75 GSTP1 (0.48) CYP1A2MAOBALDH1A1CYP2C9CYP2C19
SCHEMBL2354303 0.74 MEN1 (0.46) ALDH1A1RAB9AMEN1KMT2AKDM4E
SCHEMBL1003683 0.74 TRPV3 (0.43) CYP1A2MAOBTRPV3ALDH1A1CYP2C9
SCHEMBL144673 0.73 CYP1A2 (0.53) CYP1A2ALDH1A1CYP2C9NOTUMRAB9A
SCHEMBL3558552 0.72 KDM4E (0.66) KMOCYP1A2CYP3A4CYP2C8TGFBR1
SCHEMBL3103824 0.72 NOTUM (0.43) KMOCYP1A2CYP3A4CYP2C8TGFBR1
SCHEMBL30745584 0.72 NOTUM (0.43) KMOCYP1A2CYP3A4CYP2C8TGFBR1
Hydrochloric Acid SCHEMBL28736083 0.72 CYP1A2 (0.52) CYP1A2ALDH1A1CYP2C9NOTUMRAB9A
SCHEMBL7210200 0.72 MAPK1 (0.50) CYP1A2CYP3A4CYP2C9CYP2C19RAB9A
SCHEMBL3577075 0.71 C1R (0.44) CYP1A2CYP3A4TGFBR1TRPV3NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1021185-A4 DIDHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMA CORP (US) 2005-09-07 EP disclosed
EP-1021185-A1 DIDHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMACEUTICAL CORPORATION (US) 2000-07-26 EP disclosed
WO-1997042956-A1 DIDHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMACEUTICAL CORPORATION (US) 1997-11-20 WO disclosed