SCHEMBL6201151

SCHEMBL6201151

C[C@H](NC(=O)Oc1c(CN2CCn3cccc3C2=O)c(-c2ccccc2)nc2ccc(F)cc12)C1CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 11/20 0.45
TACR3 P29371 11/20 0.45
OPRM1 P35372 5/20 0.44
NTRK1 P04629 1/20 0.36
IDO1 P14902 2/20 0.36
MAPT P10636 1/20 0.36
TRPV4 Q9HBA0 2/20 0.35
MAPK1 P28482 1/20 0.35
DHODH Q02127 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5447117 0.90 TACR2 (0.55) TACR2TACR3OPRM1IDO1TRPV4
SCHEMBL5746603 0.83 TACR2 (0.52) TACR2TACR3OPRM1NTRK1IDO1
SCHEMBL5442143 0.82 TACR2 (0.66) TACR2TACR3OPRM1TRPV4CYP2C9
SCHEMBL5744608 0.81 TACR2 (0.55) TACR2TACR3OPRM1NTRK1TRPV4
SCHEMBL5747216 0.80 TACR2 (0.54) TACR2TACR3OPRM1NTRK1TRPV4
SCHEMBL6201232 0.80 TACR3 (0.46) TACR2TACR3OPRM1NTRK1IDO1
SCHEMBL5744442 0.79 TACR2 (0.47) TACR2TACR3OPRM1NTRK1MAPT
SCHEMBL6200585 0.79 TACR2 (0.47) TACR2TACR3OPRM1NTRK1MAPT
SCHEMBL5454432 0.77 DHODH (0.54) DHODH
SCHEMBL6249567 0.76 TACR2 (0.46) TACR2TACR3OPRM1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377567-B1 QUINOLINE-4-CARBOXAMIDE DERIVATIVES AS NK-3 AND NK-2 RECEPTOR ANTAGONISTS GLAXOSMITHKLINE SPA (IT) 2005-12-21 EP claimed