SCHEMBL6201232

SCHEMBL6201232

C[C@H](NC(=O)Oc1c(CN(C)C)c(-c2ccccc2)nc2ccc(F)cc12)C1CCCCC1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 13/20 0.46
TACR2 P21452 10/20 0.46
OPRM1 P35372 5/20 0.46
NTRK1 P04629 1/20 0.43
IDO1 P14902 2/20 0.42
DHODH Q02127 2/20 0.41
MAPK1 P28482 1/20 0.41
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6201095 0.90 TACR3 (0.54) TACR3TACR2OPRM1NTRK1
SCHEMBL5744608 0.84 TACR2 (0.55) TACR3TACR2OPRM1NTRK1
SCHEMBL5747216 0.82 TACR2 (0.54) TACR3TACR2OPRM1NTRK1
SCHEMBL6200585 0.81 TACR2 (0.47) TACR3TACR2OPRM1NTRK1MAPK1
SCHEMBL5746603 0.81 TACR2 (0.52) TACR3TACR2OPRM1NTRK1IDO1
SCHEMBL6201151 0.80 TACR2 (0.45) TACR3TACR2OPRM1NTRK1IDO1
SCHEMBL6199463 0.78 TACR3 (0.49) TACR3TACR2OPRM1NTRK1
SCHEMBL6792050 0.77 CYP2C9 (0.60) TACR3TACR2OPRM1DHODH
SCHEMBL5744442 0.77 TACR2 (0.47) TACR3TACR2OPRM1NTRK1MAPK1
SCHEMBL6249567 0.77 TACR2 (0.46) TACR3TACR2OPRM1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377567-B1 QUINOLINE-4-CARBOXAMIDE DERIVATIVES AS NK-3 AND NK-2 RECEPTOR ANTAGONISTS GLAXOSMITHKLINE SPA (IT) 2005-12-21 EP claimed