SCHEMBL6201156

SCHEMBL6201156

Brc1ccc(Br)nc1.COC(=O)c1ccc(Br)cn1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.57
KDM4E B2RXH2 5/20 0.53
ALDH1A1 P00352 2/20 0.53
L3MBTL1 Q9Y468 2/20 0.46
MAPT P10636 3/20 0.44
TP53 P04637 1/20 0.44
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
DYRK1A Q13627 1/20 0.40
CYP1A2 P05177 2/20 0.40
GAA P10253 1/20 0.40
RECQL P46063 1/20 0.40
LCK P06239 1/20 0.40
TSHR P16473 1/20 0.40
HTT P42858 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.39
GABRP O00591 1/20 0.38
GABRD O14764 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30978460 0.93 MAPK1 (0.65) MAPK1KDM4EALDH1A1L3MBTL1MAPT
SCHEMBL109364 0.93 MAPK1 (0.65) MAPK1KDM4EALDH1A1L3MBTL1MAPT
SCHEMBL30271936 0.77 MAPK1 (0.52) MAPK1KDM4EALDH1A1L3MBTL1MAPT
SCHEMBL2134366 0.77 MAPK1 (0.52) MAPK1KDM4EALDH1A1L3MBTL1MAPT
SCHEMBL15932170 0.76 KDM4E (0.56) MAPK1KDM4EALDH1A1L3MBTL1MAPT
SCHEMBL29568623 0.75 MAPK1 (0.65) MAPK1KDM4EALDH1A1L3MBTL1MAPT
SCHEMBL28049209 0.75 KDM4E (0.60) MAPK1KDM4EALDH1A1L3MBTL1NPC1
SCHEMBL28020808 0.75 KDM4E (0.60) MAPK1KDM4EALDH1A1L3MBTL1NPC1
SCHEMBL424411 0.75 MAPK1 (0.65) MAPK1KDM4EALDH1A1L3MBTL1MAPT
SCHEMBL31407736 0.75 KDM4E (0.55) MAPK1KDM4EALDH1A1SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1603885-A1 FUSED TRI AND TETRA-CYCLIC PYRAZOLE KINASE INHIBITORS Abbott Laboratories (US) 2005-12-14 EP disclosed
WO-2004080973-A1 FUSED TRI AND TETRA-CYCLIC PYRAZOLE KINASE INHIBITORS ABBOTT LABORATORIES (US) 2004-09-23 WO disclosed