SCHEMBL6201267

SCHEMBL6201267

Oc1c(Cl)ccc(CNc2ncc3nn[nH]c3n2)c1O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.33
ALOX12 P18054 1/20 0.33
HDAC3 O15379 3/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC2 Q92769 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
GFER P55789 2/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
HIF1A Q16665 1/20 0.32
CLK1 P49759 1/20 0.31
CLK2 P49760 1/20 0.31
DYRK1A Q13627 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
DYRK1B Q9Y463 1/20 0.31
RPS6KB1 P23443 1/20 0.31
NTRK1 P04629 1/20 0.30
IGF1R P08069 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6201274 0.84 CLK1 (0.34) ATMHDAC3HDAC1HDAC2HDAC6
SCHEMBL3445561 0.72 CDK2 (0.44)
SCHEMBL3443972 0.71 CCNE1 (0.38)
SCHEMBL6202539 0.71 HDAC3 (0.41) ALOX12HDAC3HDAC1HDAC2HDAC6
SCHEMBL3445213 0.70 CDK2 (0.46) HIF1ACLK1CLK2DYRK1ACLK4
SCHEMBL3445282 0.70 CDK1 (0.44) MEN1KMT2AMAPTHIF1ACLK1
SCHEMBL3444293 0.69 CDK2 (0.45)
SCHEMBL3443990 0.68 CDK2 (0.45) MEN1KMT2AMAPTHIF1ACLK1
SCHEMBL10644217 0.67 EGFR (0.39) MAPT
SCHEMBL3445563 0.67 CDK2 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed