SCHEMBL6202539

SCHEMBL6202539

COc1cc(O)c(CNc2ncc3nn[nH]c3n2)cc1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.41
HDAC1 Q13547 3/20 0.41
HDAC2 Q92769 3/20 0.41
HDAC6 Q9UBN7 3/20 0.41
GAA P10253 4/20 0.39
LMNA P02545 2/20 0.39
NPC1 O15118 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
RAB9A P51151 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
NFKB1 P19838 1/20 0.39
HTT P42858 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
EGFR P00533 2/20 0.37
ABL1 P00519 1/20 0.36
SRC P12931 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6202545 0.85 HDAC3 (0.36) HDAC3HDAC1HDAC2HDAC6GAA
SCHEMBL6203471 0.77 CCNB2 (0.46) GAALMNANPC1ALDH1A1MAPT
SCHEMBL6203475 0.73 SMN1; SMN2 (0.45) GAALMNANPC1ALDH1A1MAPT
SCHEMBL3444368 0.73 CDK2 (0.41) CCNB2CDK1CCNB1CCNB3
SCHEMBL3445017 0.72 SYK (0.36) EGFRCCNB2CDK1CCNB1CCNB3
SCHEMBL6201267 0.71 ATM (0.33) HDAC3HDAC1HDAC2HDAC6GAA
SCHEMBL3445342 0.71 CDK1 (0.44) MAPTRAB9AKDM4ECCNB2CDK1
SCHEMBL3445669 0.71 CDK2 (0.49) LMNAALDH1A1RAB9ANFKB1SMN1; SMN2
SCHEMBL3444387 0.69 CDK2 (0.49) CDK1CCNB1
SCHEMBL3444371 0.69 CDK2 (0.36) MAPTEGFRCCNB2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed